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For: Nocentini A, Supuran CT, Winum JY. Benzoxaborole compounds for therapeutic uses: a patent review (2010- 2018). Expert Opin Ther Pat. 2018;28:493-504. [PMID: 29727210 DOI: 10.1080/13543776.2018.1473379] [Cited by in Crossref: 69] [Cited by in F6Publishing: 61] [Article Influence: 13.8] [Reference Citation Analysis]
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13 Adamczyk-Woźniak A, Tarkowska M, Lazar Z, Kaczorowska E, Madura ID, Maria Dąbrowska A, Lipok J, Wieczorek D. Synthesis, structure, properties and antimicrobial activity of para trifluoromethyl phenylboronic derivatives. Bioorg Chem 2021;119:105560. [PMID: 34942467 DOI: 10.1016/j.bioorg.2021.105560] [Cited by in Crossref: 2] [Cited by in F6Publishing: 2] [Article Influence: 1.0] [Reference Citation Analysis]
14 Luo J, Jia X, Hu Y, Chen J, Sun T. Transition-metal-free, one-pot synthesis of benzoxaboroles from o-bromobenzaldehydes via visible-light-promoted borylation. Org Biomol Chem 2021;19:10455-9. [PMID: 34817493 DOI: 10.1039/d1ob01853a] [Cited by in F6Publishing: 1] [Reference Citation Analysis]
15 Kaczorowska E, Adamczyk-woźniak A, Żukowska GZ, Kostecka P, Sporzyński A. Vibrational Properties of Benzoxaboroles and Their Interactions with Candida albicans’ LeuRS. Symmetry 2021;13:1845. [DOI: 10.3390/sym13101845] [Cited by in Crossref: 2] [Cited by in F6Publishing: 2] [Article Influence: 1.0] [Reference Citation Analysis]
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17 Xiao YC, Chen XP, Deng J, Yan YH, Zhu KR, Li G, Yu JL, Brem J, Chen F, Schofield CJ, Li GB. Design and enantioselective synthesis of 3-(α-acrylic acid) benzoxaboroles to combat carbapenemase resistance. Chem Commun (Camb) 2021;57:7709-12. [PMID: 34259249 DOI: 10.1039/d1cc03026d] [Cited by in Crossref: 8] [Cited by in F6Publishing: 8] [Article Influence: 4.0] [Reference Citation Analysis]
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19 Wang X, Mohammad IS, Fan L, Zhao Z, Nurunnabi M, Sallam MA, Wu J, Chen Z, Yin L, He W. Delivery strategies of amphotericin B for invasive fungal infections. Acta Pharm Sin B 2021;11:2585-604. [PMID: 34522599 DOI: 10.1016/j.apsb.2021.04.010] [Cited by in Crossref: 12] [Cited by in F6Publishing: 13] [Article Influence: 6.0] [Reference Citation Analysis]
20 Pacholak P, Krajewska J, Wińska P, Dunikowska J, Gogowska U, Mierzejewska J, Durka K, Woźniak K, Laudy AE, Luliński S. Development of structurally extended benzosiloxaboroles - synthesis and in vitro biological evaluation. RSC Adv 2021;11:25104-21. [PMID: 35478884 DOI: 10.1039/d1ra04127d] [Cited by in Crossref: 2] [Cited by in F6Publishing: 2] [Article Influence: 1.0] [Reference Citation Analysis]
21 Nocentini A, Angeli A, Carta F, Winum JY, Zalubovskis R, Carradori S, Capasso C, Donald WA, Supuran CT. Reconsidering anion inhibitors in the general context of drug design studies of modulators of activity of the classical enzyme carbonic anhydrase. J Enzyme Inhib Med Chem 2021;36:561-80. [PMID: 33615947 DOI: 10.1080/14756366.2021.1882453] [Cited by in Crossref: 34] [Cited by in F6Publishing: 44] [Article Influence: 17.0] [Reference Citation Analysis]
22 Yan Y, Li Z, Ning X, Deng J, Yu J, Luo Y, Wang Z, Li G, Li G, Xiao Y. Discovery of 3-aryl substituted benzoxaboroles as broad-spectrum inhibitors of serine- and metallo-β-lactamases. Bioorganic & Medicinal Chemistry Letters 2021;41:127956. [DOI: 10.1016/j.bmcl.2021.127956] [Cited by in Crossref: 8] [Cited by in F6Publishing: 8] [Article Influence: 4.0] [Reference Citation Analysis]
23 Coghi PS, Zhu Y, Xie H, Hosmane NS, Zhang Y. Organoboron Compounds: Effective Antibacterial and Antiparasitic Agents. Molecules 2021;26:3309. [PMID: 34072937 DOI: 10.3390/molecules26113309] [Cited by in Crossref: 7] [Cited by in F6Publishing: 7] [Article Influence: 3.5] [Reference Citation Analysis]
24 Soydan E, Olcay AC, Bilir G, Taş Ö, Şentürk M, Ekinci D, Supuran CT. Investigation of pesticides on honey bee carbonic anhydrase inhibition. J Enzyme Inhib Med Chem 2020;35:1923-7. [PMID: 33078633 DOI: 10.1080/14756366.2020.1835885] [Cited by in Crossref: 2] [Cited by in F6Publishing: 3] [Article Influence: 1.0] [Reference Citation Analysis]
25 Nocentini A, Hewitt CS, Mastrolorenzo MD, Flaherty DP, Supuran CT. Anion inhibition studies of the α-carbonic anhydrases from Neisseria gonorrhoeae. J Enzyme Inhib Med Chem 2021;36:1061-6. [PMID: 34030562 DOI: 10.1080/14756366.2021.1929202] [Cited by in Crossref: 2] [Cited by in F6Publishing: 3] [Article Influence: 1.0] [Reference Citation Analysis]
26 Zhao J, Chen J, Xu Q, Li H. Synthesis of Benzoxaboroles by ortho-Oxalkylation of Arylboronic Acids with Aldehydes/Ketones in the Presence of Brønsted Acids. Org Lett 2021;23:1986-90. [PMID: 33646001 DOI: 10.1021/acs.orglett.1c00032] [Cited by in Crossref: 3] [Cited by in F6Publishing: 3] [Article Influence: 1.5] [Reference Citation Analysis]
27 Kwon MH, Lee DY, Kang HE. Development and Validation of an LC-MS/MS Method for Quantification of the Novel Antibacterial Candidate DA-7010 in Plasma and Application to a Preclinical Pharmacokinetic Study. Pharmaceuticals (Basel) 2021;14:163. [PMID: 33670597 DOI: 10.3390/ph14020163] [Cited by in Crossref: 1] [Cited by in F6Publishing: 1] [Article Influence: 0.5] [Reference Citation Analysis]
28 Golovanov IS, Sukhorukov AY. Merging Boron with Nitrogen-Oxygen Bonds: A Review on BON Heterocycles. Top Curr Chem (Cham) 2021;379:8. [PMID: 33544252 DOI: 10.1007/s41061-020-00317-3] [Cited by in Crossref: 2] [Cited by in F6Publishing: 3] [Article Influence: 1.0] [Reference Citation Analysis]
29 Oguz M, Kalay E, Akocak S, Nocentini A, Lolak N, Boga M, Yilmaz M, Supuran CT. Synthesis of calix[4]azacrown substituted sulphonamides with antioxidant, acetylcholinesterase, butyrylcholinesterase, tyrosinase and carbonic anhydrase inhibitory action. J Enzyme Inhib Med Chem 2020;35:1215-23. [PMID: 32401067 DOI: 10.1080/14756366.2020.1765166] [Cited by in Crossref: 15] [Cited by in F6Publishing: 11] [Article Influence: 7.5] [Reference Citation Analysis]
30 Vega-valdez IR, Rosalez NM, Santiago-Quintana M, Farfán-García ED, Marvin A. Soriano-Ursúa. Docking Simulations Exhibit Bortezomib and other Boron-containing Peptidomimetics as Potential Inhibitors of SARS-CoV-2 Main Protease. CCB 2021;14:279-88. [DOI: 10.2174/2212796814999201102195651] [Cited by in Crossref: 6] [Cited by in F6Publishing: 6] [Article Influence: 3.0] [Reference Citation Analysis]
31 Estevez-Fregoso E, Farfán-García ED, García-Coronel IH, Martínez-Herrera E, Alatorre A, Scorei RI, Soriano-Ursúa MA. Effects of boron-containing compounds in the fungal kingdom. J Trace Elem Med Biol 2021;65:126714. [PMID: 33453473 DOI: 10.1016/j.jtemb.2021.126714] [Cited by in Crossref: 3] [Cited by in F6Publishing: 3] [Article Influence: 1.5] [Reference Citation Analysis]
32 Goyal N, Patel M, Batra S. Modern Drug Discovery and Development in the Area of Leishmaniasis. Drug Discovery and Drug Development 2021. [DOI: 10.1007/978-981-15-8002-4_5] [Cited by in Crossref: 2] [Article Influence: 1.0] [Reference Citation Analysis]
33 Supuran CT. A Story on Carbon Dioxide and Its Hydration. New Trends in Macromolecular and Supramolecular Chemistry for Biological Applications 2021. [DOI: 10.1007/978-3-030-57456-7_6] [Reference Citation Analysis]
34 Vermelho AB, Mori M, Donald WA, Supuran CT. Challenges and Promises for Obtaining New Antiprotozoal Drugs: What’s Going Wrong? Topics in Medicinal Chemistry 2021. [DOI: 10.1007/7355_2021_136] [Cited by in Crossref: 1] [Cited by in F6Publishing: 1] [Article Influence: 0.5] [Reference Citation Analysis]
35 Nocentini A, Vermelho AB, Supuran CT. Targeting Carbonic Anhydrases from Trypanosoma cruzi and Leishmania spp. as a Therapeutic Strategy to Obtain New Antiprotozoal Drugs. Topics in Medicinal Chemistry 2021. [DOI: 10.1007/7355_2021_140] [Cited by in Crossref: 1] [Article Influence: 0.5] [Reference Citation Analysis]
36 Supuran CT. Carbonic Anhydrase Inhibitors: Designing Isozyme-Specific Inhibitors as Therapeutic Agents. Progress in Drug Research 2021. [DOI: 10.1007/978-3-030-79511-5_10] [Reference Citation Analysis]
37 Rotella DP. Heterocycles in drug discovery: Properties and preparation. Advances in Heterocyclic Chemistry 2021. [DOI: 10.1016/bs.aihch.2020.10.002] [Cited by in Crossref: 4] [Cited by in F6Publishing: 5] [Article Influence: 2.0] [Reference Citation Analysis]
38 Küçükbay H, Gönül Z, Küçükbay FZ, Angeli A, Bartolucci G, Supuran CT. Preparation, carbonic anhydrase enzyme inhibition and antioxidant activity of novel 7-amino-3,4-dihydroquinolin-2(1H)-one derivatives incorporating mono or dipeptide moiety. J Enzyme Inhib Med Chem 2020;35:1021-6. [PMID: 32297533 DOI: 10.1080/14756366.2020.1751620] [Cited by in Crossref: 5] [Cited by in F6Publishing: 5] [Article Influence: 1.7] [Reference Citation Analysis]
39 Niemczyk E, Pogrzeba J, Adamczyk-Woźniak A, Lipok J. Boronic Acids of Pharmaceutical Importance Affect the Growth and Photosynthetic Apparatus of Cyanobacteria in a Dose-Dependent Manner. Toxins (Basel) 2020;12:E793. [PMID: 33322165 DOI: 10.3390/toxins12120793] [Cited by in Crossref: 1] [Cited by in F6Publishing: 1] [Article Influence: 0.3] [Reference Citation Analysis]
40 Bonardi A, Nocentini A, Cadoni R, Del Prete S, Dumy P, Capasso C, Gratteri P, Supuran CT, Winum JY. Benzoxaboroles: New Potent Inhibitors of the Carbonic Anhydrases of the Pathogenic Bacterium Vibrio cholerae. ACS Med Chem Lett 2020;11:2277-84. [PMID: 33214840 DOI: 10.1021/acsmedchemlett.0c00403] [Cited by in Crossref: 11] [Cited by in F6Publishing: 12] [Article Influence: 3.7] [Reference Citation Analysis]
41 Giordani F, Paape D, Vincent IM, Pountain AW, Fernández-Cortés F, Rico E, Zhang N, Morrison LJ, Freund Y, Witty MJ, Peter R, Edwards DY, Wilkes JM, van der Hooft JJJ, Regnault C, Read KD, Horn D, Field MC, Barrett MP. Veterinary trypanocidal benzoxaboroles are peptidase-activated prodrugs. PLoS Pathog 2020;16:e1008932. [PMID: 33141865 DOI: 10.1371/journal.ppat.1008932] [Cited by in Crossref: 9] [Cited by in F6Publishing: 9] [Article Influence: 3.0] [Reference Citation Analysis]
42 Umumararungu T, Mukazayire MJ, Mpenda M, Mukanyangezi MF, Nkuranga JB, Mukiza J, Olawode EO. A review of recent advances in anti-tubercular drug development. Indian J Tuberc 2020;67:539-59. [PMID: 33077057 DOI: 10.1016/j.ijtb.2020.07.017] [Cited by in Crossref: 4] [Cited by in F6Publishing: 4] [Article Influence: 1.3] [Reference Citation Analysis]
43 Angeli A, Carta F, Nocentini A, Winum JY, Zalubovskis R, Akdemir A, Onnis V, Eldehna WM, Capasso C, Simone G, Monti SM, Carradori S, Donald WA, Dedhar S, Supuran CT. Carbonic Anhydrase Inhibitors Targeting Metabolism and Tumor Microenvironment. Metabolites 2020;10:E412. [PMID: 33066524 DOI: 10.3390/metabo10100412] [Cited by in Crossref: 57] [Cited by in F6Publishing: 70] [Article Influence: 19.0] [Reference Citation Analysis]
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45 Liu RJ, Long T, Li H, Zhao J, Li J, Wang M, Palencia A, Lin J, Cusack S, Wang ED. Molecular basis of the multifaceted functions of human leucyl-tRNA synthetase in protein synthesis and beyond. Nucleic Acids Res 2020;48:4946-59. [PMID: 32232361 DOI: 10.1093/nar/gkaa189] [Cited by in Crossref: 7] [Cited by in F6Publishing: 7] [Article Influence: 2.3] [Reference Citation Analysis]
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48 Ćwik P, Ciosek-Skibińska P, Zabadaj M, Luliński S, Durka K, Wróblewski W. Differential Sensing of Saccharides Based on an Array of Fluorinated Benzosiloxaborole Receptors. Sensors (Basel) 2020;20:E3540. [PMID: 32580489 DOI: 10.3390/s20123540] [Cited by in Crossref: 2] [Cited by in F6Publishing: 2] [Article Influence: 0.7] [Reference Citation Analysis]
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51 Li X, Wu S, Dong G, Chen S, Ma Z, Liu D, Sheng C. Natural Product Evodiamine with Borate Trigger Unit: Discovery of Potent Antitumor Agents against Colon Cancer. ACS Med Chem Lett 2020;11:439-44. [PMID: 32292547 DOI: 10.1021/acsmedchemlett.9b00513] [Cited by in Crossref: 13] [Cited by in F6Publishing: 14] [Article Influence: 4.3] [Reference Citation Analysis]
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57 Walker AL, Denis A, Bingham RP, Bouillot A, Edgar EV, Ferrie A, Holmes DS, Laroze A, Liddle J, Fouchet M, Moquette A, Nassau P, Pearce AC, Polyakova O, Smith KJ, Thomas P, Thorpe JH, Trottet L, Wang Y, Hovnanian A. Design and development of a series of borocycles as selective, covalent kallikrein 5 inhibitors. Bioorganic & Medicinal Chemistry Letters 2019;29:126675. [DOI: 10.1016/j.bmcl.2019.126675] [Cited by in Crossref: 5] [Cited by in F6Publishing: 5] [Article Influence: 1.3] [Reference Citation Analysis]
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59 Larcher A, Nocentini A, Supuran CT, Winum JY, van der Lee A, Vasseur JJ, Laurencin D, Smietana M. Bis-benzoxaboroles: Design, Synthesis, and Biological Evaluation as Carbonic Anhydrase Inhibitors. ACS Med Chem Lett 2019;10:1205-10. [PMID: 31413806 DOI: 10.1021/acsmedchemlett.9b00252] [Cited by in Crossref: 12] [Cited by in F6Publishing: 12] [Article Influence: 3.0] [Reference Citation Analysis]
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