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For: Johnson BM, Shu YZ, Zhuo X, Meanwell NA. Metabolic and Pharmaceutical Aspects of Fluorinated Compounds. J Med Chem 2020;63:6315-86. [PMID: 32182061 DOI: 10.1021/acs.jmedchem.9b01877] [Cited by in Crossref: 82] [Cited by in F6Publishing: 53] [Article Influence: 41.0] [Reference Citation Analysis]
Number Citing Articles
1 Fang Y, Li X, Liu C, Tang J, Chen Z. Nucleophilic Substitution of Selenosulfonates with Me3SiCF2Br: Facile and Efficient Access to Bromodifluoromethylated Selenides under Metal-Free Conditions. J Org Chem 2021;86:18081-93. [PMID: 34823360 DOI: 10.1021/acs.joc.1c02349] [Reference Citation Analysis]
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3 Cheng J, Zhang H, Lv J, Zheng J. Palladium‐Catalyzed Intermolecular Dicarbofunctionalization of Unactivated Alkenes: Synthesis of Fluoroalkylated Heterocycles with All‐Carbon Quaternary Centers. European J Organic Chem 2022;2022. [DOI: 10.1002/ejoc.202101342] [Reference Citation Analysis]
4 Sorrentino JP, Altman RA. Fluoroalkylation of Dextromethorphan Improves CNS Exposure and Metabolic Stability. ACS Med Chem Lett . [DOI: 10.1021/acsmedchemlett.2c00055] [Reference Citation Analysis]
5 Saranya PV, Aneeja T, Anilkumar G. Palladium‐catalyzed difluoromethylation and difluoroalkylation reactions: An overview. Appl Organomet Chem. [DOI: 10.1002/aoc.6503] [Reference Citation Analysis]
6 Grychowska K, Olejarz-maciej A, Blicharz K, Pietruś W, Karcz T, Kurczab R, Koczurkiewicz P, Doroz-płonka A, Latacz G, Keeri AR, Piska K, Satała G, Pęgiel J, Trybała W, Jastrzębska-więsek M, Bojarski AJ, Lamaty F, Partyka A, Walczak M, Krawczyk M, Malikowska-racia N, Popik P, Zajdel P. Overcoming undesirable hERG affinity by incorporating fluorine atoms: A case of MAO-B inhibitors derived from 1 H-pyrrolo-[3,2-c]quinolines. European Journal of Medicinal Chemistry 2022. [DOI: 10.1016/j.ejmech.2022.114329] [Reference Citation Analysis]
7 Wang C, Wang L, Meng Q, Huang Z, Ma N, Wang C. Crystal structure of ( E )-2-((3-fluoropyridin-4-yl)methylene)-7-methoxy-3,4-dihydronaphthalen-1(2 H )-one, C 17 H 14 FNO 2. Zeitschrift für Kristallographie - New Crystal Structures 2021;236:1073-5. [DOI: 10.1515/ncrs-2021-0223] [Reference Citation Analysis]
8 Gopalsamy A, Aulabaugh AE, Barakat A, Beaumont KC, Cabral S, Canterbury DP, Casimiro-Garcia A, Chang JS, Chen MZ, Choi C, Dow RL, Fadeyi OO, Feng X, France SP, Howard RM, Janz JM, Jasti J, Jasuja R, Jones LH, King-Ahmad A, Knee KM, Kohrt JT, Limberakis C, Liras S, Martinez CA, McClure KF, Narayanan A, Narula J, Novak JJ, O'Connell TN, Parikh MD, Piotrowski DW, Plotnikova O, Robinson RP, Sahasrabudhe PV, Sharma R, Thuma BA, Vasa D, Wei L, Wenzel AZ, Withka JM, Xiao J, Yayla HG. PF-07059013: A Noncovalent Modulator of Hemoglobin for Treatment of Sickle Cell Disease. J Med Chem 2021;64:326-42. [PMID: 33356244 DOI: 10.1021/acs.jmedchem.0c01518] [Cited by in Crossref: 3] [Cited by in F6Publishing: 3] [Article Influence: 1.5] [Reference Citation Analysis]
9 Schmidhammer H, Erli F, Guerrieri E, Spetea M. Development of Diphenethylamines as Selective Kappa Opioid Receptor Ligands and Their Pharmacological Activities. Molecules 2020;25:E5092. [PMID: 33147885 DOI: 10.3390/molecules25215092] [Reference Citation Analysis]
10 Liu Y, Uras G, Onuwaje I, Li W, Yao H, Xu S, Li X, Li X, Phillips J, Allen S, Gong Q, Zhang H, Zhu Z, Liu J, Xu J. Novel inhibitors of AChE and Aβ aggregation with neuroprotective properties as lead compounds for the treatment of Alzheimer's disease. European Journal of Medicinal Chemistry 2022. [DOI: 10.1016/j.ejmech.2022.114305] [Reference Citation Analysis]
11 Han Z, Zhang C. Fluorination and Fluoroalkylation Reactions Mediated by Hypervalent Iodine Reagents. Adv Synth Catal 2020;362:4256-92. [DOI: 10.1002/adsc.202000750] [Cited by in Crossref: 17] [Cited by in F6Publishing: 8] [Article Influence: 8.5] [Reference Citation Analysis]
12 Panish R, Thieu T, Balsells J. Copper-Catalyzed Synthesis of 5-Carboxyl-4-perfluoroalkyl Triazoles. Org Lett 2021;23:5937-41. [PMID: 34286985 DOI: 10.1021/acs.orglett.1c02037] [Reference Citation Analysis]
13 Tong CL, Xu XH, Qing FL. Nucleophilic and Radical Heptafluoroisopropoxylation with Redox-Active Reagents. Angew Chem Int Ed Engl 2021;60:22915-24. [PMID: 34414643 DOI: 10.1002/anie.202109572] [Reference Citation Analysis]
14 Li Y, Wang Y, Ye Z, Zhang S, Ye X, Yuan Z. Trifluoromethyl Selenoxides: Electrophilic Reagents for C-H Trifluoromethylselenolation of (Hetero)Arene. Org Lett 2022. [PMID: 35436121 DOI: 10.1021/acs.orglett.2c00916] [Reference Citation Analysis]
15 Mondal R, Agbaria M, Nairoukh Z. Fluorinated Rings: Conformation and Application. Chemistry 2021;27:7193-213. [PMID: 33512034 DOI: 10.1002/chem.202005425] [Cited by in Crossref: 5] [Cited by in F6Publishing: 4] [Article Influence: 5.0] [Reference Citation Analysis]
16 Zafrani Y, Parvari G, Amir D, Ghindes-Azaria L, Elias S, Pevzner A, Fridkin G, Berliner A, Gershonov E, Eichen Y, Saphier S, Katalan S. Modulation of the H-Bond Basicity of Functional Groups by α-Fluorine-Containing Functions and its Implications for Lipophilicity and Bioisosterism. J Med Chem 2021;64:4516-31. [PMID: 33844540 DOI: 10.1021/acs.jmedchem.0c01868] [Cited by in Crossref: 1] [Cited by in F6Publishing: 1] [Article Influence: 1.0] [Reference Citation Analysis]
17 Abula A, Xu Z, Zhu Z, Peng C, Chen Z, Zhu W, Aisa HA. Substitution Effect of the Trifluoromethyl Group on the Bioactivity in Medicinal Chemistry: Statistical Analysis and Energy Calculations. J Chem Inf Model 2020;60:6242-50. [DOI: 10.1021/acs.jcim.0c00898] [Cited by in Crossref: 2] [Cited by in F6Publishing: 2] [Article Influence: 1.0] [Reference Citation Analysis]
18 Wen Z, Salmaso V, Jung YH, Phung NB, Gopinatth V, Shah Q, Patterson AT, Randle JCR, Chen Z, Salvemini D, Lieberman DI, Whitehead GS, Karcz TP, Cook DN, Jacobson KA. Bridged Piperidine Analogues of a High Affinity Naphthalene-Based P2Y14R Antagonist. J Med Chem 2022. [PMID: 35113556 DOI: 10.1021/acs.jmedchem.1c01964] [Reference Citation Analysis]
19 Tosstorff A, Cole JC, Taylor R, Harris SF, Kuhn B. Identification of Noncompetitive Protein–Ligand Interactions for Structural Optimization. J Chem Inf Model 2020;60:6595-611. [DOI: 10.1021/acs.jcim.0c00858] [Cited by in Crossref: 4] [Cited by in F6Publishing: 3] [Article Influence: 2.0] [Reference Citation Analysis]
20 Heard DM, Doobary S, Lennox AJJ. 3D Printed Reactionware for Synthetic Electrochemistry with Hydrogen Fluoride Reagents. ChemElectroChem 2021;8:2070-4. [DOI: 10.1002/celc.202100496] [Cited by in Crossref: 2] [Cited by in F6Publishing: 1] [Article Influence: 2.0] [Reference Citation Analysis]
21 Lloyd MD, Yevglevskis M, Nathubhai A, James TD, Threadgill MD, Woodman TJ. Racemases and epimerases operating through a 1,1-proton transfer mechanism: reactivity, mechanism and inhibition. Chem Soc Rev 2021;50:5952-84. [PMID: 34027955 DOI: 10.1039/d0cs00540a] [Cited by in Crossref: 1] [Cited by in F6Publishing: 1] [Article Influence: 1.0] [Reference Citation Analysis]
22 Fu J, Tsapy Takia IR, Chen P, Liu W, Jiang C, Yao W, Zeng X, Wang Y, Han X. Synthesis of 2-chromanone-fused [3.2.0] bicycles through a phosphine-mediated tandem [3 + 2] cyclization/intramolecular Wittig reaction. Org Chem Front 2021;8:6323-9. [DOI: 10.1039/d1qo01013a] [Reference Citation Analysis]
23 Pal S, Chandra G, Patel S, Singh S. Fluorinated Nucleosides: Synthesis, Modulation in Conformation and Therapeutic Application. Chem Rec 2022;:e202100335. [PMID: 35253973 DOI: 10.1002/tcr.202100335] [Reference Citation Analysis]
24 Bhutani P, Joshi G, Raja N, Bachhav N, Rajanna PK, Bhutani H, Paul AT, Kumar R. U.S. FDA Approved Drugs from 2015-June 2020: A Perspective. J Med Chem 2021;64:2339-81. [PMID: 33617716 DOI: 10.1021/acs.jmedchem.0c01786] [Cited by in Crossref: 18] [Cited by in F6Publishing: 8] [Article Influence: 18.0] [Reference Citation Analysis]
25 Piscelli BA, Sanders W, Yu C, Al Maharik N, Lebl T, Cormanich RA, O'Hagan D. Fluorine-Induced Pseudo-Anomeric Effects in Methoxycyclohexanes through Electrostatic 1,3-Diaxial Interactions. Chemistry 2020;26:11989-94. [PMID: 32588927 DOI: 10.1002/chem.202003058] [Cited by in Crossref: 2] [Cited by in F6Publishing: 2] [Article Influence: 1.0] [Reference Citation Analysis]
26 Boudreau MW, Mulligan MP, Shapiro DJ, Fan TM, Hergenrother PJ. Activators of the Anticipatory Unfolded Protein Response with Enhanced Selectivity for Estrogen Receptor Positive Breast Cancer. J Med Chem 2022. [PMID: 35080871 DOI: 10.1021/acs.jmedchem.1c01730] [Reference Citation Analysis]
27 de Gonzalo G, Alcántara AR. Recent Developments in the Synthesis of β-Diketones. Pharmaceuticals (Basel) 2021;14:1043. [PMID: 34681266 DOI: 10.3390/ph14101043] [Reference Citation Analysis]
28 Grollier K, Taponard A, De Zordo-Banliat A, Magnier E, Billard T. Metal-free nucleophilic trifluoromethylselenolation via an iodide-mediated umpolung reactivity of trifluoromethylselenotoluenesulfonate. Beilstein J Org Chem 2020;16:3032-7. [PMID: 33363671 DOI: 10.3762/bjoc.16.252] [Cited by in Crossref: 1] [Cited by in F6Publishing: 1] [Article Influence: 0.5] [Reference Citation Analysis]
29 Grollier K, Chefdeville E, De Zordo-banliat A, Pegot B, Dagousset G, Magnier E, Billard T. Fe-mediated nucleophilic trifluoromethylselenolation of activated alkyl bromides via umpolung reactivity of trifluoromethyl tolueneselenosulfinate. Tetrahedron 2021;100:132498. [DOI: 10.1016/j.tet.2021.132498] [Reference Citation Analysis]
30 Cong W, Sun Y, Sun YF, Yan WB, Zhang YL, Gao ZF, Wang CH, Hou GG, Zhang JJ. Trifluoromethyl-substituted 3,5-bis(arylidene)-4-piperidones as potential anti-hepatoma and anti-inflammation agents by inhibiting NF-кB activation. J Enzyme Inhib Med Chem 2021;36:1622-31. [PMID: 34284695 DOI: 10.1080/14756366.2021.1953996] [Reference Citation Analysis]
31 Wen S, Tian Q, Chen Y, Zhang Y, Cheng G. Annulation of CF3-Imidoyl Sulfoxonium Ylides with 1,3-Dicarbonyl Compounds: Access to 1,2,3-Trisubstituted 5-Trifluoromethylpyrroles. Org Lett 2021;23:7407-11. [PMID: 34543038 DOI: 10.1021/acs.orglett.1c02598] [Cited by in Crossref: 2] [Cited by in F6Publishing: 1] [Article Influence: 2.0] [Reference Citation Analysis]
32 Casa S, Henary M. Synthesis and Applications of Selected Fluorine-Containing Fluorophores. Molecules 2021;26:1160. [PMID: 33671600 DOI: 10.3390/molecules26041160] [Cited by in F6Publishing: 1] [Reference Citation Analysis]
33 Varga B, Tóth BL, Béke F, Csenki JT, Kotschy A, Novák Z. Synthesis and Photochemical Application of Hydrofluoroolefin (HFO) Based Fluoroalkyl Building Block. Org Lett 2021;23:4925-9. [PMID: 34097412 DOI: 10.1021/acs.orglett.1c01709] [Cited by in Crossref: 1] [Article Influence: 1.0] [Reference Citation Analysis]
34 Wen S, Chen Y, Tian Q, Zhang Y, Cheng G. Transition-Metal-, Additive-, and Solvent-Free [3 + 3] Annulation of RCF2-Imidoyl Sulfoxonium Ylides with Cyclopropenones to Give Multifunctionalized CF3-Pyridones. J Org Chem 2021. [PMID: 34965129 DOI: 10.1021/acs.joc.1c02464] [Reference Citation Analysis]
35 Morand S, Jubault P, Bouillon JP, Couve-Bonnaire S. gem-Heteroatom-Substituted Fluoroalkenes as Mimics of Amide Derivatives or Phosphates: A Comprehensive Review. Chemistry 2021;27:17273-92. [PMID: 34533868 DOI: 10.1002/chem.202102548] [Cited by in Crossref: 1] [Article Influence: 1.0] [Reference Citation Analysis]
36 Troelsen NS, Clausen MH. Library Design Strategies To Accelerate Fragment‐Based Drug Discovery. Chem Eur J 2020;26:11391-403. [DOI: 10.1002/chem.202000584] [Cited by in Crossref: 6] [Cited by in F6Publishing: 5] [Article Influence: 3.0] [Reference Citation Analysis]
37 Liu L, Ran L, Gu Y, Zhang C. Facile synthesis of selenocarbamyl fluorides, selenoureas and their derivatives with [Me 4 N][SeCF 3 ]. Org Chem Front 2021;8:5736-43. [DOI: 10.1039/d1qo00736j] [Reference Citation Analysis]
38 Kittilä T, Calero P, Fredslund F, Lowe PT, Tezé D, Nieto-Domínguez M, O'Hagan D, Nikel PI, Welner DH. Oligomerization engineering of the fluorinase enzyme leads to an active trimer that supports synthesis of fluorometabolites in vitro. Microb Biotechnol 2022. [PMID: 35084776 DOI: 10.1111/1751-7915.14009] [Reference Citation Analysis]
39 Grollier K, De Zordo‐banliat A, Bourdreux F, Pegot B, Dagousset G, Magnier E, Billard T. (Trifluoromethylselenyl)methylchalcogenyl as Emerging Fluorinated Groups: Synthesis under Photoredox Catalysis and Determination of the Lipophilicity. Chem Eur J 2021;27:6028-33. [DOI: 10.1002/chem.202100053] [Cited by in Crossref: 6] [Cited by in F6Publishing: 1] [Article Influence: 6.0] [Reference Citation Analysis]
40 Lee W, Lee Y, Yoo M, Han SB, Kim HJ. Photoredox-catalyzed halotrifluoromethylations of alkynes with triethylammonium halides: synthesis of tetrasubstituted alkenes containing CF 3 and halogens. Org Chem Front 2020;7:3209-14. [DOI: 10.1039/d0qo00893a] [Cited by in Crossref: 4] [Article Influence: 2.0] [Reference Citation Analysis]
41 Gao Y, Wan X, Feng Z, Fang L, Chen X, Jia Y, Tian M. The influence of fluorine terminal group and flexible spacers on properties of the liquid crystal dimers. Liquid Crystals 2022;49:380-91. [DOI: 10.1080/02678292.2021.1970837] [Reference Citation Analysis]
42 Li J, Xi W, Zhong R, Yang J, Wang L, Ding H, Wang Z. HFIP-catalyzed direct dehydroxydifluoroalkylation of benzylic and allylic alcohols with difluoroenoxysilanes. Chem Commun 2021;57:1050-3. [DOI: 10.1039/d0cc06980a] [Cited by in Crossref: 4] [Article Influence: 4.0] [Reference Citation Analysis]
43 Ruyet L, Lapuh MI, Koshti VS, Földesi T, Jubault P, Poisson T, Novák Z, Besset T. Z-Selective Pd-catalyzed 2,2,2-trifluoroethylation of acrylamides at room temperature. Chem Commun (Camb) 2021;57:6241-4. [PMID: 34079967 DOI: 10.1039/d1cc02007b] [Cited by in Crossref: 3] [Article Influence: 3.0] [Reference Citation Analysis]
44 Zhang JQ, Hu D, Song J, Ren H. [3 + 2]-Annulation of gem-Difluoroalkenes and Pyridinium Ylides: Access to Functionalized 2-Fluoroindolizines. J Org Chem 2021;86:4646-60. [PMID: 33683121 DOI: 10.1021/acs.joc.0c03041] [Cited by in Crossref: 1] [Article Influence: 1.0] [Reference Citation Analysis]
45 Politanskaya L, Tretyakov E, Xi C. Synthesis of polyfluorinated 4‑hydroxyquinolin-2(1H)‑ones based on the cyclization of 2-alkynylanilines with carbon dioxide. Journal of Fluorine Chemistry 2021;242:109720. [DOI: 10.1016/j.jfluchem.2020.109720] [Cited by in Crossref: 2] [Article Influence: 2.0] [Reference Citation Analysis]
46 Spetea M, Schmidhammer H. Kappa Opioid Receptor Ligands and Pharmacology: Diphenethylamines, a Class of Structurally Distinct, Selective Kappa Opioid Ligands. Handb Exp Pharmacol 2021. [PMID: 33454858 DOI: 10.1007/164_2020_431] [Reference Citation Analysis]
47 Yang J, Liu S, Hong P, Li J, Wang Z, Ren J. Synthesis of 2,2-Difluoro-3-hydroxy-1,4-diketones via an HFIP-Catalyzed Mukaiyama Aldol Reaction of Glyoxal Monohydrates with Difluoroenoxysilanes. J Org Chem 2022;87:1144-53. [PMID: 34994195 DOI: 10.1021/acs.joc.1c02504] [Cited by in Crossref: 2] [Cited by in F6Publishing: 2] [Article Influence: 2.0] [Reference Citation Analysis]
48 Chen XQ, Lu H, Chen CX, Zeng R, Wang DY, Shi CY, Zhang A. Palladium-Catalyzed gem-Difluoroallylation Reaction between Aryltributyltin and Bromodifluoromethylated Alkenes. J Org Chem 2022. [PMID: 35075894 DOI: 10.1021/acs.joc.1c02800] [Reference Citation Analysis]
49 Meyer DN, Cortés González MA, Jiang X, Johansson-Holm L, Pourghasemi Lati M, Elgland M, Nordeman P, Antoni G, Szabó KJ. Base-catalysed 18F-labelling of trifluoromethyl ketones. Application to the synthesis of 18F-labelled neutrophil elastase inhibitors. Chem Commun (Camb) 2021;57:8476-9. [PMID: 34346419 DOI: 10.1039/d1cc03624f] [Cited by in Crossref: 1] [Cited by in F6Publishing: 1] [Article Influence: 1.0] [Reference Citation Analysis]
50 Schiesser S, Chepliaka H, Kollback J, Quennesson T, Czechtizky W, Cox RJ. N -Trifluoromethyl Amines and Azoles: An Underexplored Functional Group in the Medicinal Chemist’s Toolbox. J Med Chem 2020;63:13076-89. [DOI: 10.1021/acs.jmedchem.0c01457] [Cited by in Crossref: 4] [Cited by in F6Publishing: 3] [Article Influence: 2.0] [Reference Citation Analysis]
51 Edilova YO, Kudyakova YS, Kiskin MA, Burgart YV, Saloutin VI, Bazhin DN. Expanding 1,2,4-triketone toolbox for use as fluorinated building blocks in the synthesis of pyrazoles, pyridazinones and β-diketohydrazones. Journal of Fluorine Chemistry 2022;253:109932. [DOI: 10.1016/j.jfluchem.2021.109932] [Reference Citation Analysis]
52 Zhao Y, Wang X, Yao R, Li C, Xu Z, Zhang L, Han G, Hou J, Liu Y, Song Y. Iron‐Catalyzed Alkene Trifluoromethylation in Tandem with Phenol Dearomatizing Spirocyclization: Regioselective Construction of Trifluoromethylated Spirocarbocycles. Adv Synth Catal 2022;364:637-42. [DOI: 10.1002/adsc.202101201] [Reference Citation Analysis]
53 Modak A, Alegre-Requena JV, de Lescure L, Rynders KJ, Paton RS, Race NJ. Homologation of Electron-Rich Benzyl Bromide Derivatives via Diazo C-C Bond Insertion. J Am Chem Soc 2021. [PMID: 34898193 DOI: 10.1021/jacs.1c11503] [Reference Citation Analysis]
54 Gao H, Lin S, Zhang S, Chen W, Liu X, Yang G, Lerner RA, Xu H, Zhou Z, Yi W. gem ‐Difluoromethylene Alkyne‐Enabled Diverse C−H Functionalization and Application to the on‐DNA Synthesis of Difluorinated Isocoumarins. Angew Chem Int Ed 2021;60:1959-66. [DOI: 10.1002/anie.202013052] [Cited by in Crossref: 12] [Cited by in F6Publishing: 8] [Article Influence: 6.0] [Reference Citation Analysis]
55 Csenki JT, Mészáros Á, Gonda Z, Novák Z. Stereoselective Direct N-Trifluoropropenylation of Heterocycles with a Hypervalent Iodonium Reagent. Chemistry 2021;27:15638-43. [PMID: 34549840 DOI: 10.1002/chem.202102840] [Reference Citation Analysis]
56 Li Y, Li X, Li X, Shi D. Highly E-Selective Synthesis of α-Fluoro-β-arylalkenyl Sulfones from gem-Difluoroalkenes with Sodium Sulfinates. J Org Chem 2021;86:6983-93. [PMID: 33852316 DOI: 10.1021/acs.joc.1c00490] [Cited by in Crossref: 2] [Article Influence: 2.0] [Reference Citation Analysis]
57 Wang H, Dong J, Shi J, Zhang C. Trifluoromethylselenolation reactions using the versatile [Me4N][SeCF3] reagent. Tetrahedron 2021;99:132476. [DOI: 10.1016/j.tet.2021.132476] [Cited by in Crossref: 1] [Cited by in F6Publishing: 1] [Article Influence: 1.0] [Reference Citation Analysis]
58 Adamik R, Földesi T, Novák Z. Photocatalytic Palladium-Catalyzed Fluoroalkylation of Styrene Derivatives. Org Lett 2020;22:8091-5. [PMID: 33001655 DOI: 10.1021/acs.orglett.0c03043] [Cited by in Crossref: 5] [Cited by in F6Publishing: 1] [Article Influence: 2.5] [Reference Citation Analysis]
59 Yang L, Zhang Y, Deng J, Ma A, Zhang X, Zhang S, Peng J. Oxidative [3+2] Annulation of Pyridinium Salts with gem ‐Difluoroalkenes: Synthesis of 2‐Fluoroindolizines. Asian J Org Chem 2021;10:1679-82. [DOI: 10.1002/ajoc.202100253] [Cited by in Crossref: 1] [Cited by in F6Publishing: 1] [Article Influence: 1.0] [Reference Citation Analysis]
60 Espitia Cogollo E, Jios E, Hidalgo A, Ulic SE, Echeverría GA, Piro OE, Jios JL. The Bonding Interactions in Fluorinated Vinylogous Amides: A CF 3 ‐Substituted Carbonyl‐β‐Aminoenone as a Case Study. Crystal Research and Technology 2021;56:2000162. [DOI: 10.1002/crat.202000162] [Reference Citation Analysis]
61 Yang L, Zhang CP. Revisiting the Balz-Schiemann Reaction of Aryldiazonium Tetrafluoroborate in Different Solvents under Catalyst- and Additive-Free Conditions. ACS Omega 2021;6:21595-603. [PMID: 34471763 DOI: 10.1021/acsomega.1c02825] [Reference Citation Analysis]
62 St-Gelais J, Côté É, Lainé D, Johnson PA, Giguère D. Addressing the Structural Complexity of Fluorinated Glucose Analogues: Insight into Lipophilicities and Solvation Effects. Chemistry 2020;26:13499-506. [PMID: 32652740 DOI: 10.1002/chem.202002825] [Cited by in Crossref: 9] [Cited by in F6Publishing: 6] [Article Influence: 4.5] [Reference Citation Analysis]
63 Potenti S, Spada L, Fusè M, Mancini G, Gualandi A, Leonardi C, Cozzi PG, Puzzarini C, Barone V. 4-Fluoro-Threonine: From Diastereoselective Synthesis to pH-Dependent Conformational Equilibrium in Aqueous Solution. ACS Omega 2021;6:13170-81. [PMID: 34056467 DOI: 10.1021/acsomega.1c01007] [Cited by in Crossref: 1] [Article Influence: 1.0] [Reference Citation Analysis]
64 Tóth BL, Sályi G, Domján A, Egyed O, Bényei A, Gonda Z, Novák Z. Z ‐Selective Fluoroalkenylation of (Hetero)Aromatic Systems by Iodonium Reagents in Palladium‐Catalyzed Directed C−H Activation. Adv Synth Catal 2022;364:348-54. [DOI: 10.1002/adsc.202101108] [Reference Citation Analysis]
65 Schmid JC, Frey K, Scheiner M, Garzón JFG, Stafforst L, Fricke JN, Schuppe M, Schiewe H, Zeeck A, Weber T, Usón I, Kemkemer R, Decker M, Grond S. The Structure of Cyclodecatriene Collinolactone, its Biosynthesis, and Semisynthetic Analogues: Effects of Monoastral Phenotype and Protection from Intracellular Oxidative Stress. Angew Chem Int Ed Engl 2021;60:23212-6. [PMID: 34415670 DOI: 10.1002/anie.202106802] [Reference Citation Analysis]
66 Tan KL, Wang HN, Dong T, Zhang CP. Trifluoromethylselenolation and N-acylation of indoles with [Me4N][SeCF3]. Org Biomol Chem 2021;19:5368-76. [PMID: 34047751 DOI: 10.1039/d1ob00842k] [Cited by in Crossref: 2] [Article Influence: 2.0] [Reference Citation Analysis]
67 Li C, Zhao Y, Zhou J, Wang X, Hou J, Song Y, Liu W, Han G. Synthesis of difluoroalkylated 2-azaspiro[4.5]decane derivatives via copper-catalyzed difluoroalkylation/dearomatization of N -benzylacrylamides. Org Biomol Chem 2020;18:8376-80. [DOI: 10.1039/d0ob01833c] [Cited by in Crossref: 2] [Article Influence: 1.0] [Reference Citation Analysis]
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