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For: Teixeira C, Vale N, Pérez B, Gomes A, Gomes JR, Gomes P. "Recycling" classical drugs for malaria. Chem Rev 2014;114:11164-220. [PMID: 25329927 DOI: 10.1021/cr500123g] [Cited by in Crossref: 80] [Cited by in F6Publishing: 62] [Article Influence: 10.0] [Reference Citation Analysis]
Number Citing Articles
1 Srinivasarao K, Agarwal P, Srivastava K, Haq W, Puri SK, Katti SB. Design, synthesis, and in vitro antiplasmodial activity of 4-aminoquinolines containing modified amino acid conjugates. Med Chem Res 2016;25:1148-62. [DOI: 10.1007/s00044-016-1555-5] [Cited by in Crossref: 8] [Cited by in F6Publishing: 5] [Article Influence: 1.3] [Reference Citation Analysis]
2 Fonte M, Tassi N, Fontinha D, Bouzón-Arnáiz I, Ferraz R, Araújo MJ, Fernàndez-Busquets X, Prudêncio M, Gomes P, Teixeira C. 4,9-Diaminoacridines and 4-Aminoacridines as Dual-Stage Antiplasmodial Hits. ChemMedChem 2021;16:788-92. [PMID: 33217195 DOI: 10.1002/cmdc.202000740] [Cited by in Crossref: 1] [Cited by in F6Publishing: 1] [Article Influence: 0.5] [Reference Citation Analysis]
3 Beus M, Rajić Z, Maysinger D, Mlinarić Z, Antunović M, Marijanović I, Fontinha D, Prudêncio M, Held J, Olgen S, Zorc B. SAHAquines, Novel Hybrids Based on SAHA and Primaquine Motifs, as Potential Cytostatic and Antiplasmodial Agents. ChemistryOpen 2018;7:624-38. [PMID: 30151334 DOI: 10.1002/open.201800117] [Cited by in Crossref: 8] [Cited by in F6Publishing: 10] [Article Influence: 2.0] [Reference Citation Analysis]
4 C S Pinheiro L, M Feitosa L, O Gandi M, F Silveira F, Boechat N. The Development of Novel Compounds Against Malaria: Quinolines, Triazolpyridines, Pyrazolopyridines and Pyrazolopyrimidines. Molecules 2019;24:E4095. [PMID: 31766184 DOI: 10.3390/molecules24224095] [Cited by in Crossref: 17] [Cited by in F6Publishing: 9] [Article Influence: 5.7] [Reference Citation Analysis]
5 Çapcı A, Lorion MM, Wang H, Simon N, Leidenberger M, Borges silva MC, Moreira DRM, Zhu Y, Meng Y, Chen JY, Lee YM, Friedrich O, Kappes B, Wang J, Ackermann L, Tsogoeva SB. Artemisinin–(Iso)quinoline Hybrids by C−H Activation and Click Chemistry: Combating Multidrug‐Resistant Malaria. Angew Chem 2019;131:13200-13. [DOI: 10.1002/ange.201907224] [Cited by in Crossref: 4] [Cited by in F6Publishing: 2] [Article Influence: 1.3] [Reference Citation Analysis]
6 Van de Walle T, Cools L, Mangelinckx S, D'hooghe M. Recent contributions of quinolines to antimalarial and anticancer drug discovery research. Eur J Med Chem 2021;226:113865. [PMID: 34655985 DOI: 10.1016/j.ejmech.2021.113865] [Cited by in Crossref: 1] [Article Influence: 1.0] [Reference Citation Analysis]
7 Silva AT, Lobo L, Oliveira IS, Gomes J, Teixeira C, Nogueira F, Marques EF, Ferraz R, Gomes P. Building on Surface-Active Ionic Liquids for the Rescuing of the Antimalarial Drug Chloroquine. Int J Mol Sci 2020;21:E5334. [PMID: 32727096 DOI: 10.3390/ijms21155334] [Cited by in Crossref: 2] [Cited by in F6Publishing: 2] [Article Influence: 1.0] [Reference Citation Analysis]
8 Garbacz M, Stecko S. Synthesis of chiral branched allylamines through dual photoredox/nickel catalysis. Org Biomol Chem 2021;19:8578-85. [PMID: 34553201 DOI: 10.1039/d1ob01624e] [Reference Citation Analysis]
9 Gomes A, Fernandes I, Teixeira C, Mateus N, Sottomayor MJ, Gomes P. A Quinacrine Analogue Selective Against Gastric Cancer Cells: Insight from Biochemical and Biophysical Studies. ChemMedChem 2016;11:2703-12. [PMID: 27863116 DOI: 10.1002/cmdc.201600477] [Cited by in Crossref: 8] [Cited by in F6Publishing: 6] [Article Influence: 1.3] [Reference Citation Analysis]
10 Bento CM, Gomes MS, Silva T. Looking beyond Typical Treatments for Atypical Mycobacteria. Antibiotics (Basel) 2020;9:E18. [PMID: 31947883 DOI: 10.3390/antibiotics9010018] [Cited by in Crossref: 10] [Cited by in F6Publishing: 10] [Article Influence: 5.0] [Reference Citation Analysis]
11 Fonte M, Tassi N, Gomes P, Teixeira C. Acridine-Based Antimalarials-From the Very First Synthetic Antimalarial to Recent Developments. Molecules 2021;26:600. [PMID: 33498868 DOI: 10.3390/molecules26030600] [Cited by in Crossref: 1] [Cited by in F6Publishing: 1] [Article Influence: 1.0] [Reference Citation Analysis]
12 Silva AT, Oliveira IS, Gomes J, Aguiar L, Fontinha D, Duarte D, Nogueira F, Prudêncio M, Marques EF, Teixeira C, Ferraz R, Gomes P. Drug-Derived Surface-Active Ionic Liquids: A Cost-Effective Way To Expressively Increase the Blood-Stage Antimalarial Activity of Primaquine. ChemMedChem 2021;:e202100650. [PMID: 34882979 DOI: 10.1002/cmdc.202100650] [Reference Citation Analysis]
13 Pinheiro LC, Feitosa LM, Silveira FFD, Boechat N. Current Antimalarial Therapies and Advances in the Development of Semi-Synthetic Artemisinin Derivatives. An Acad Bras Ciênc 2018;90:1251-71. [DOI: 10.1590/0001-3765201820170830] [Cited by in Crossref: 22] [Cited by in F6Publishing: 17] [Article Influence: 5.5] [Reference Citation Analysis]
14 Neelarapu R, Maignan JR, Lichorowic CL, Monastyrskyi A, Mutka TS, LaCrue AN, Blake LD, Casandra D, Mashkouri S, Burrows JN, Willis PA, Kyle DE, Manetsch R. Design and Synthesis of Orally Bioavailable Piperazine Substituted 4(1H)-Quinolones with Potent Antimalarial Activity: Structure-Activity and Structure-Property Relationship Studies. J Med Chem 2018;61:1450-73. [PMID: 29215279 DOI: 10.1021/acs.jmedchem.7b00738] [Cited by in Crossref: 12] [Cited by in F6Publishing: 12] [Article Influence: 3.0] [Reference Citation Analysis]
15 Maurya SS, Bahuguna A, Khan SI, Kumar D, Kholiya R, Rawat DS. N-Substituted aminoquinoline-pyrimidine hybrids: Synthesis, in vitro antimalarial activity evaluation and docking studies. Eur J Med Chem 2019;162:277-89. [PMID: 30448417 DOI: 10.1016/j.ejmech.2018.11.021] [Cited by in Crossref: 12] [Cited by in F6Publishing: 8] [Article Influence: 3.0] [Reference Citation Analysis]
16 Mu W, Wang M, Li H, Huang D, Zhang Y, Li C, Liu Y, Wu Y. Palladium-Catalyzed Regioselective Oxidative Annulation of Cyclohexanones and 2-Aminophenyl Ketones Using Molecular Oxygen as the Sole Oxidant. Adv Synth Catal 2017;359:4250-7. [DOI: 10.1002/adsc.201700715] [Cited by in Crossref: 13] [Cited by in F6Publishing: 6] [Article Influence: 2.6] [Reference Citation Analysis]
17 Vale N, Aguiar L, Gomes P. Antimicrobial peptides: a new class of antimalarial drugs? Front Pharmacol 2014;5:275. [PMID: 25566072 DOI: 10.3389/fphar.2014.00275] [Cited by in Crossref: 36] [Cited by in F6Publishing: 34] [Article Influence: 4.5] [Reference Citation Analysis]
18 Gomes A, Machado M, Lobo L, Nogueira F, Prudêncio M, Teixeira C, Gomes P. N-Cinnamoylation of Antimalarial Classics: Effects of Using Acyl Groups Other than Cinnamoyl toward Dual-Stage Antimalarials. ChemMedChem 2015;10:1344-9. [PMID: 26038181 DOI: 10.1002/cmdc.201500164] [Cited by in Crossref: 11] [Cited by in F6Publishing: 11] [Article Influence: 1.6] [Reference Citation Analysis]
19 Bhagat S, Arfeen M, Das G, Ramkumar M, Khan SI, Tekwani BL, Bharatam PV. Design, synthesis and biological evaluation of 4-aminoquinoline-guanylthiourea derivatives as antimalarial agents. Bioorg Chem 2019;91:103094. [PMID: 31376783 DOI: 10.1016/j.bioorg.2019.103094] [Cited by in Crossref: 7] [Cited by in F6Publishing: 4] [Article Influence: 2.3] [Reference Citation Analysis]
20 Dhiman S, Saini HK, Nandwana NK, Kumar D, Kumar A. Copper-catalyzed synthesis of quinoline derivatives via tandem Knoevenagel condensation, amination and cyclization. RSC Adv 2016;6:23987-94. [DOI: 10.1039/c6ra03798d] [Cited by in Crossref: 17] [Article Influence: 2.8] [Reference Citation Analysis]
21 Jain S, Kumar A, Saini D. Novel arylidene derivatives of quinoline based thiazolidinones: Synthesis, in vitro, in vivo and in silico study as antimalarials. Exp Parasitol 2018;185:107-14. [PMID: 29355497 DOI: 10.1016/j.exppara.2018.01.015] [Cited by in Crossref: 8] [Cited by in F6Publishing: 2] [Article Influence: 2.0] [Reference Citation Analysis]
22 Perković I, Raić-Malić S, Fontinha D, Prudêncio M, Pessanha de Carvalho L, Held J, Tandarić T, Vianello R, Zorc B, Rajić Z. Harmicines - harmine and cinnamic acid hybrids as novel antiplasmodial hits. Eur J Med Chem 2020;187:111927. [PMID: 31812035 DOI: 10.1016/j.ejmech.2019.111927] [Cited by in Crossref: 10] [Cited by in F6Publishing: 8] [Article Influence: 3.3] [Reference Citation Analysis]
23 Tripathi M, Taylor D, Khan SI, Tekwani BL, Ponnan P, Das US, Velpandian T, Rawat DS. Hybridization of Fluoro-amodiaquine (FAQ) with Pyrimidines: Synthesis and Antimalarial Efficacy of FAQ-Pyrimidines. ACS Med Chem Lett 2019;10:714-9. [PMID: 31097988 DOI: 10.1021/acsmedchemlett.8b00496] [Cited by in Crossref: 7] [Cited by in F6Publishing: 6] [Article Influence: 2.3] [Reference Citation Analysis]
24 Teixeira C, Ventura C, Gomes JRB, Gomes P, Martins F. Cinnamic Derivatives as Antitubercular Agents: Characterization by Quantitative Structure-Activity Relationship Studies. Molecules 2020;25:E456. [PMID: 31973244 DOI: 10.3390/molecules25030456] [Cited by in Crossref: 2] [Article Influence: 1.0] [Reference Citation Analysis]
25 Tripathi M, Khan SI, Ponnan P, Kholiya R, Rawat DS. Aminoquinoline-Pyrimidine-Modified Anilines: Synthesis, In Vitro Antiplasmodial Activity, Cytotoxicity, Mechanistic Studies and ADME Predictions. ChemistrySelect 2017;2:9074-83. [DOI: 10.1002/slct.201701558] [Cited by in Crossref: 3] [Cited by in F6Publishing: 1] [Article Influence: 0.6] [Reference Citation Analysis]
26 Bhanot A, Sundriyal S. Physicochemical Profiling and Comparison of Research Antiplasmodials and Advanced Stage Antimalarials with Oral Drugs. ACS Omega 2021;6:6424-37. [PMID: 33718733 DOI: 10.1021/acsomega.1c00104] [Reference Citation Analysis]
27 Gopinath P, Yadav RK, Shukla PK, Srivastava K, Puri SK, Muraleedharan KM. Broad spectrum anti-infective properties of benzisothiazolones and the parallels in their anti-bacterial and anti-fungal effects. Bioorg Med Chem Lett 2017;27:1291-5. [PMID: 28159413 DOI: 10.1016/j.bmcl.2017.01.027] [Cited by in Crossref: 7] [Cited by in F6Publishing: 6] [Article Influence: 1.4] [Reference Citation Analysis]
28 Gurskaya LY, Belyanskaya DS, Ryabukhin DS, Nilov DI, Boyarskaya IA, Vasilyev AV. Reactions of N,3-diarylpropiolamides with arenes under superelectrophilic activation: synthesis of 4,4-diaryl-3,4-dihydroquinolin-2(1H)-ones and their derivatives. Beilstein J Org Chem 2016;12:950-6. [PMID: 27340485 DOI: 10.3762/bjoc.12.93] [Cited by in Crossref: 7] [Article Influence: 1.2] [Reference Citation Analysis]
29 Dembitsky VM, Ermolenko E, Savidov N, Gloriozova TA, Poroikov VV. Antiprotozoal and Antitumor Activity of Natural Polycyclic Endoperoxides: Origin, Structures and Biological Activity. Molecules 2021;26:686. [PMID: 33525706 DOI: 10.3390/molecules26030686] [Cited by in Crossref: 2] [Cited by in F6Publishing: 2] [Article Influence: 2.0] [Reference Citation Analysis]
30 Silva TB, Bernardino AM, Ferreira MDLG, Rogerio KR, Carvalho LJ, Boechat N, Pinheiro LC. Design, synthesis and anti-P. falciparum activity of pyrazolopyridine–sulfonamide derivatives. Bioorganic & Medicinal Chemistry 2016;24:4492-8. [DOI: 10.1016/j.bmc.2016.07.049] [Cited by in Crossref: 24] [Cited by in F6Publishing: 18] [Article Influence: 4.0] [Reference Citation Analysis]
31 Rajić KPZ, Mlinarić Z, Uzelac L, Kralj M, Zorc B. Chloroquine Urea Derivatives: Synthesis and Antitumor Activity in Vitro. Acta Pharm 2018;68:471-83. [PMID: 31259711 DOI: 10.2478/acph-2018-0039] [Cited by in Crossref: 4] [Cited by in F6Publishing: 3] [Article Influence: 1.3] [Reference Citation Analysis]
32 Chopin N, Iikawa S, Bosson J, Lavoignat A, Bonnot G, Bienvenu A, Picot S, Bouillon J, Médebielle M. 7-Chloro-4-aminoquinoline γ-hydroxy-γ-lactam derived-tetramates as a new family of antimalarial compounds. Bioorganic & Medicinal Chemistry Letters 2016;26:5308-11. [DOI: 10.1016/j.bmcl.2016.09.038] [Cited by in Crossref: 3] [Cited by in F6Publishing: 3] [Article Influence: 0.5] [Reference Citation Analysis]
33 Ghosh C, Chaubey S, Tatu U, Haldar J. Aryl-alkyl-lysines: small molecular membrane-active antiplasmodial agents. Medchemcomm 2017;8:434-9. [PMID: 30108761 DOI: 10.1039/c6md00589f] [Cited by in Crossref: 4] [Cited by in F6Publishing: 3] [Article Influence: 0.7] [Reference Citation Analysis]
34 Aguiar L, Machado M, Sanches-Vaz M, Prudêncio M, Vale N, Gomes P. Coupling the cell-penetrating peptides transportan and transportan 10 to primaquine enhances its activity against liver-stage malaria parasites. Medchemcomm 2019;10:221-6. [PMID: 30881610 DOI: 10.1039/c8md00447a] [Cited by in Crossref: 10] [Cited by in F6Publishing: 6] [Article Influence: 2.5] [Reference Citation Analysis]
35 Lacerda AF, Pelegrini PB, de Oliveira DM, Vasconcelos ÉA, Grossi-de-Sá MF. Anti-parasitic Peptides from Arthropods and their Application in Drug Therapy. Front Microbiol 2016;7:91. [PMID: 26903970 DOI: 10.3389/fmicb.2016.00091] [Cited by in Crossref: 22] [Cited by in F6Publishing: 22] [Article Influence: 3.7] [Reference Citation Analysis]
36 Liu ZQ. Enhancing Antioxidant Effect against Peroxyl Radical-Induced Oxidation of DNA: Linking with Ferrocene Moiety! Chem Rec 2019;19:2385-97. [PMID: 30946536 DOI: 10.1002/tcr.201800201] [Cited by in Crossref: 4] [Cited by in F6Publishing: 2] [Article Influence: 1.3] [Reference Citation Analysis]
37 Pereira FM, de Oliveira AR, Mattioli MP, Carneiro FT. Diagnosis and Treatment of Plasmodium Infection in Captive Black and White Tegus. J Comp Pathol 2021;183:9-12. [PMID: 33714436 DOI: 10.1016/j.jcpa.2020.12.006] [Reference Citation Analysis]
38 Silveira FF, Feitosa LM, Mafra JCM, Ferreira MDLG, Rogerio KR, Carvalho LJM, Boechat N, Pinheiro LCS. Synthesis and anti-Plasmodium falciparum evaluation of novel pyrazolopyrimidine derivatives. Med Chem Res 2018;27:1876-84. [DOI: 10.1007/s00044-018-2199-4] [Cited by in Crossref: 3] [Cited by in F6Publishing: 1] [Article Influence: 0.8] [Reference Citation Analysis]
39 Gomes A, Ferraz R, Ficker L, Collins MS, Prudêncio C, Cushion MT, Teixeira C, Gomes P. Chloroquine Analogues as Leads against Pneumocystis Lung Pathogens. Antimicrob Agents Chemother 2018;62:e00983-18. [PMID: 30201816 DOI: 10.1128/AAC.00983-18] [Cited by in Crossref: 4] [Cited by in F6Publishing: 2] [Article Influence: 1.0] [Reference Citation Analysis]
40 Ye X, Xu B, Sun J, Dai L, Shao Y, Zhang Y, Chen J. Pd-Catalyzed Approach for Assembling 9-Arylacridines via a Cascade Tandem Reaction of 2-(Arylamino)benzonitrile with Arylboronic Acids in Water. J Org Chem 2020;85:13004-14. [PMID: 32957780 DOI: 10.1021/acs.joc.0c01654] [Cited by in Crossref: 1] [Cited by in F6Publishing: 1] [Article Influence: 0.5] [Reference Citation Analysis]
41 Shi L, Pan L, Li Y, Liu Q. Copper(II)-Catalyzed Aerobic Oxidative Desulfitative 6π Electrocyclization: Efficient Synthesis of Diverse 4-Aminoquinolines. Adv Synth Catal 2017;359:2457-70. [DOI: 10.1002/adsc.201700410] [Cited by in Crossref: 12] [Cited by in F6Publishing: 3] [Article Influence: 2.4] [Reference Citation Analysis]
42 Cao Z, Zhu Y, Li X, He Y, Zhang J, Xu L, Wei Y. tert-Butyl Bromide-Promoted Intramolecular Cyclization of 2-Arylamino Phenyl Ketones and Its Combination with Cu-Catalyzed C-N Coupling: Synthesis of Acridines at Room Temperature. J Org Chem 2020;85:10167-74. [PMID: 32568540 DOI: 10.1021/acs.joc.0c00137] [Cited by in Crossref: 4] [Cited by in F6Publishing: 2] [Article Influence: 2.0] [Reference Citation Analysis]
43 Witschel MC, Rottmann M, Schwab A, Leartsakulpanich U, Chitnumsub P, Seet M, Tonazzi S, Schwertz G, Stelzer F, Mietzner T, Mcnamara C, Thater F, Freymond C, Jaruwat A, Pinthong C, Riangrungroj P, Oufir M, Hamburger M, Mäser P, Sanz-alonso LM, Charman S, Wittlin S, Yuthavong Y, Chaiyen P, Diederich F. Inhibitors of Plasmodial Serine Hydroxymethyltransferase (SHMT): Cocrystal Structures of Pyrazolopyrans with Potent Blood- and Liver-Stage Activities. J Med Chem 2015;58:3117-30. [DOI: 10.1021/jm501987h] [Cited by in Crossref: 31] [Cited by in F6Publishing: 27] [Article Influence: 4.4] [Reference Citation Analysis]
44 Silva AT, Bento CM, Pena AC, Figueiredo LM, Prudêncio C, Aguiar L, Silva T, Ferraz R, Gomes MS, Teixeira C, Gomes P. Cinnamic Acid Conjugates in the Rescuing and Repurposing of Classical Antimalarial Drugs. Molecules 2019;25:E66. [PMID: 31878190 DOI: 10.3390/molecules25010066] [Cited by in Crossref: 9] [Cited by in F6Publishing: 8] [Article Influence: 3.0] [Reference Citation Analysis]
45 Rogerio KR, Graebin CS, Pinto Domingues LH, Oliveira LS, de Souza Fernandes da Silva V, Daniel-Ribeiro CT, Carvalho LJM, Boechat N. Novel Quinolinyl-pyrrolo[3,4-d]pyrimidine-2,5-dione Derivatives Against Chloroquine-resistant Plasmodium falciparum. Curr Top Med Chem 2020;20:99-110. [PMID: 31648638 DOI: 10.2174/1568026619666191019100711] [Cited by in Crossref: 2] [Article Influence: 0.7] [Reference Citation Analysis]
46 Shalini, Kumar S, Gendrot M, Fonta I, Mosnier J, Cele N, Awolade P, Singh P, Pradines B, Kumar V. Amide Tethered 4-Aminoquinoline-naphthalimide Hybrids: A New Class of Possible Dual Function Antiplasmodials. ACS Med Chem Lett 2020;11:2544-52. [PMID: 33335678 DOI: 10.1021/acsmedchemlett.0c00536] [Cited by in Crossref: 2] [Cited by in F6Publishing: 2] [Article Influence: 1.0] [Reference Citation Analysis]
47 Araujo JSC, de Souza BC, Costa Junior DB, Oliveira LDM, Santana IB, Duarte AA, Lacerda PS, dos Santos Junior MC, Leite FHA. Identification of new promising Plasmodium falciparum superoxide dismutase allosteric inhibitors through hierarchical pharmacophore-based virtual screening and molecular dynamics. J Mol Model 2018;24. [DOI: 10.1007/s00894-018-3746-0] [Cited by in Crossref: 4] [Cited by in F6Publishing: 2] [Article Influence: 1.0] [Reference Citation Analysis]
48 Bujok R, Wróbel Z, Wojciechowski K. Simple synthesis of 4-cyanoquinoline N-oxides. Tetrahedron Letters 2016;57:1014-8. [DOI: 10.1016/j.tetlet.2016.01.072] [Cited by in Crossref: 7] [Cited by in F6Publishing: 3] [Article Influence: 1.2] [Reference Citation Analysis]
49 Fonte M, Fagundes N, Gomes A, Ferraz R, Prudêncio C, Araújo MJ, Gomes P, Teixeira C. Development of a synthetic route towards N4,N9-disubstituted 4,9-diaminoacridines: On the way to multi-stage antimalarials. Tetrahedron Letters 2019;60:1166-9. [DOI: 10.1016/j.tetlet.2019.03.052] [Cited by in Crossref: 3] [Cited by in F6Publishing: 2] [Article Influence: 1.0] [Reference Citation Analysis]
50 Silva AT, Cerqueira MJ, Prudêncio C, Fernandes MH, Costa-rodrigues J, Teixeira C, Gomes P, Ferraz R. Antiproliferative Organic Salts Derived from Betulinic Acid: Disclosure of an Ionic Liquid Selective Against Lung and Liver Cancer Cells. ACS Omega 2019;4:5682-9. [DOI: 10.1021/acsomega.8b03691] [Cited by in Crossref: 7] [Cited by in F6Publishing: 1] [Article Influence: 2.3] [Reference Citation Analysis]
51 Senadi GC, Dhandabani GK, Hu W, Wang J. Metal-free annulation/aerobic oxidative dehydrogenation of cyclohexanones with o-acylanilines: efficient syntheses of acridines. Green Chem 2016;18:6241-5. [DOI: 10.1039/c6gc02396g] [Cited by in Crossref: 22] [Article Influence: 3.7] [Reference Citation Analysis]
52 Çapcı A, Lorion MM, Wang H, Simon N, Leidenberger M, Borges Silva MC, Moreira DRM, Zhu Y, Meng Y, Chen JY, Lee YM, Friedrich O, Kappes B, Wang J, Ackermann L, Tsogoeva SB. Artemisinin-(Iso)quinoline Hybrids by C-H Activation and Click Chemistry: Combating Multidrug-Resistant Malaria. Angew Chem Int Ed Engl 2019;58:13066-79. [PMID: 31290221 DOI: 10.1002/anie.201907224] [Cited by in Crossref: 42] [Cited by in F6Publishing: 34] [Article Influence: 14.0] [Reference Citation Analysis]
53 Maignan JR, Lichorowic CL, Giarrusso J, Blake LD, Casandra D, Mutka TS, Lacrue AN, Burrows JN, Willis PA, Kyle DE, Manetsch R. ICI 56,780 Optimization: Structure–Activity Relationship Studies of 7-(2-Phenoxyethoxy)-4(1 H )-quinolones with Antimalarial Activity. J Med Chem 2016;59:6943-60. [DOI: 10.1021/acs.jmedchem.6b00759] [Cited by in Crossref: 11] [Cited by in F6Publishing: 9] [Article Influence: 1.8] [Reference Citation Analysis]
54 Adebayo JO, Tijjani H, Adegunloye AP, Ishola AA, Balogun EA, Malomo SO. Enhancing the antimalarial activity of artesunate. Parasitol Res 2020;119:2749-64. [PMID: 32638101 DOI: 10.1007/s00436-020-06786-1] [Cited by in Crossref: 5] [Cited by in F6Publishing: 3] [Article Influence: 2.5] [Reference Citation Analysis]
55 Senadi GC, Hu W, Garkhedkar AM, Boominathan SSK, Wang J. Palladium( ii )-catalysed regioselective synthesis of 3,4-disubstituted quinolines and 2,3,5-trisubstituted pyrroles from alkenes via anti-Markovnikov selectivity. Chem Commun 2015;51:13795-8. [DOI: 10.1039/c5cc05196g] [Cited by in Crossref: 31] [Article Influence: 4.4] [Reference Citation Analysis]
56 Ferraz R, Noronha J, Murtinheira F, Nogueira F, Machado M, Prudêncio M, Parapini S, D'alessandro S, Teixeira C, Gomes A, Prudêncio C, Gomes P. Primaquine-based ionic liquids as a novel class of antimalarial hits. RSC Adv 2016;6:56134-8. [DOI: 10.1039/c6ra10759a] [Cited by in Crossref: 22] [Cited by in F6Publishing: 1] [Article Influence: 3.7] [Reference Citation Analysis]
57 Maurya SS, Khan SI, Bahuguna A, Kumar D, Rawat DS. Synthesis, antimalarial activity, heme binding and docking studies of N-substituted 4-aminoquinoline-pyrimidine molecular hybrids. Eur J Med Chem 2017;129:175-85. [PMID: 28222317 DOI: 10.1016/j.ejmech.2017.02.024] [Cited by in Crossref: 24] [Cited by in F6Publishing: 17] [Article Influence: 4.8] [Reference Citation Analysis]
58 Murce E, Cuya-Guizado TR, Padilla-Chavarria HI, França TCC, Pimentel AS. Structure-based de novo design, molecular docking and molecular dynamics of primaquine analogues acting as quinone reductase II inhibitors. J Mol Graph Model 2015;62:235-44. [PMID: 26521207 DOI: 10.1016/j.jmgm.2015.10.001] [Cited by in Crossref: 3] [Article Influence: 0.4] [Reference Citation Analysis]
59 Pinheiro LC, Boechat N, Ferreira Mde L, Júnior CC, Jesus AM, Leite MM, Souza NB, Krettli AU. Anti-Plasmodium falciparum activity of quinoline-sulfonamide hybrids. Bioorg Med Chem 2015;23:5979-84. [PMID: 26190461 DOI: 10.1016/j.bmc.2015.06.056] [Cited by in Crossref: 23] [Cited by in F6Publishing: 22] [Article Influence: 3.3] [Reference Citation Analysis]
60 Varela JN, Lammoglia Cobo MF, Pawar SV, Yadav VG. Cheminformatic Analysis of Antimalarial Chemical Space Illuminates Therapeutic Mechanisms and Offers Strategies for Therapy Development. J Chem Inf Model 2017;57:2119-31. [PMID: 28810125 DOI: 10.1021/acs.jcim.7b00072] [Cited by in Crossref: 3] [Cited by in F6Publishing: 3] [Article Influence: 0.6] [Reference Citation Analysis]
61 Guedes RA, Serra P, Salvador JA, Guedes RC. Computational Approaches for the Discovery of Human Proteasome Inhibitors: An Overview. Molecules 2016;21:E927. [PMID: 27438821 DOI: 10.3390/molecules21070927] [Cited by in Crossref: 13] [Cited by in F6Publishing: 11] [Article Influence: 2.2] [Reference Citation Analysis]
62 Boechat N, Carvalho RCC, Ferreira MLG, Coutinho JP, Sa PM, Seito LN, Rosas EC, Krettli AU, Bastos MM, Pinheiro LCS. Antimalarial and anti-inflammatory activities of new chloroquine and primaquine hybrids: Targeting the blockade of malaria parasite transmission. Bioorg Med Chem 2020;28:115832. [PMID: 33166927 DOI: 10.1016/j.bmc.2020.115832] [Cited by in Crossref: 1] [Cited by in F6Publishing: 2] [Article Influence: 0.5] [Reference Citation Analysis]
63 Ferraz R, Pinheiro M, Gomes A, Teixeira C, Prudêncio C, Reis S, Gomes P. Effects of novel triple-stage antimalarial ionic liquids on lipid membrane models. Bioorganic & Medicinal Chemistry Letters 2017;27:4190-3. [DOI: 10.1016/j.bmcl.2017.07.006] [Cited by in Crossref: 17] [Cited by in F6Publishing: 15] [Article Influence: 3.4] [Reference Citation Analysis]
64 Shalini, Legac J, Adeniyi AA, Kisten P, Rosenthal PJ, Singh P, Kumar V. Functionalized Naphthalimide-4-aminoquinoline Conjugates as Promising Antiplasmodials, with Mechanistic Insights. ACS Med Chem Lett 2020;11:154-61. [PMID: 32071682 DOI: 10.1021/acsmedchemlett.9b00521] [Cited by in Crossref: 6] [Cited by in F6Publishing: 5] [Article Influence: 3.0] [Reference Citation Analysis]
65 Lau S, Galván A, Merchant RR, Battilocchio C, Souto JA, Berry MB, Ley SV. Machines vs Malaria: A Flow-Based Preparation of the Drug Candidate OZ439. Org Lett 2015;17:3218-21. [DOI: 10.1021/acs.orglett.5b01307] [Cited by in Crossref: 37] [Cited by in F6Publishing: 26] [Article Influence: 5.3] [Reference Citation Analysis]
66 Korotchenko V, Sathunuru R, Gerena L, Caridha D, Li Q, Kreishman-Deitrick M, Smith PL, Lin AJ. Antimalarial activity of 4-amidinoquinoline and 10-amidinobenzonaphthyridine derivatives. J Med Chem 2015;58:3411-31. [PMID: 25654185 DOI: 10.1021/jm501809x] [Cited by in Crossref: 15] [Cited by in F6Publishing: 12] [Article Influence: 2.1] [Reference Citation Analysis]