| 1 |
Xu Y, Fan H, Yang F, Xu S, Zhao X, Liao X, Zhang X. PPh(3)-Mediated Cascade Reaction of 2-Alkynylnitrobenzenes and Thioureas for the Construction of Imidazo[4,5-b]indole-2-thiones. J Org Chem 2023;88:2801-8. [PMID: 36800292 DOI: 10.1021/acs.joc.2c02434] [Reference Citation Analysis]
|
| 2 |
Rajesab P, Chavan PW, Badiger JG, C Hanamshetty P. MULTICOMPONENT ONE-POT SYNTHESIS OF NOVEL INDOLE ANALOGUES AS POTENT ANTIOXIDANT AGENTS. Asian J Pharm Clin Res 2022. [DOI: 10.22159/ajpcr.2022.v15i6.43926] [Reference Citation Analysis]
|
| 3 |
Arjunan V, Devi GD. Structure, conformations, vibrations and quantum chemical investigations of 2–(1H–indol–3–yl)–2–oxoacetic acid. Journal of Molecular Structure 2022;1256:132570. [DOI: 10.1016/j.molstruc.2022.132570] [Reference Citation Analysis]
|
| 4 |
Setia Budi H, Fakri Mustafa Y, Al-hamdani MM, Surendar A, Ramezani M. Synthesis of heterocycles from propargylamines. Synthetic Communications 2021;51:3694-716. [DOI: 10.1080/00397911.2021.2001660] [Cited by in Crossref: 2] [Cited by in F6Publishing: 2] [Article Influence: 1.0] [Reference Citation Analysis]
|
| 5 |
Hu X, Xie X, Gan Y, Wang G, Liu Y. Nickel-Catalyzed β-Regioselective Amination/Cyclization of Ynamide-Nitriles with Amines: Synthesis of Functionalized 3-Aminoindoles and 4-Aminoisoquinolines. Org Lett 2021;23:1296-301. [PMID: 33533626 DOI: 10.1021/acs.orglett.0c04278] [Cited by in Crossref: 7] [Cited by in F6Publishing: 7] [Article Influence: 3.5] [Reference Citation Analysis]
|
| 6 |
Hu X, Tan Z, Liu Z, Chen F, Jiang H, Zeng W. Rh( iii )-Catalyzed sulfonylamination of α-indolyl alcohols via Csp 2 –Csp 3 bond cleavage. Org Chem Front 2021;8:983-7. [DOI: 10.1039/d0qo01426e] [Cited by in Crossref: 3] [Cited by in F6Publishing: 3] [Article Influence: 1.5] [Reference Citation Analysis]
|
| 7 |
Chen W, Li K, Liao W, Liang W, Qiu P, Liang C, Su G, Mo D. An iron(iii)-catalyzed dehydrogenative cross-coupling reaction of indoles with benzylamines to prepare 3-aminoindole derivatives. Green Chem 2021;23:9610-9616. [DOI: 10.1039/d1gc02849a] [Cited by in Crossref: 1] [Cited by in F6Publishing: 1] [Article Influence: 0.5] [Reference Citation Analysis]
|
| 8 |
Srinivas S, Neeraja P, Banothu V, Kumar Dubey P, Mukkanti K, Pal S. Synthesis, Biological Evaluation and In silico Studies of Compounds Based on Tryptophan‐Naproxen‐Triazole Hybrids. ChemistrySelect 2020;5:14741-14746. [DOI: 10.1002/slct.202003786] [Cited by in Crossref: 2] [Cited by in F6Publishing: 3] [Article Influence: 0.7] [Reference Citation Analysis]
|
| 9 |
Akuamoah DA, Opoku E, Tia R, Adei E. 1,3-Dipolar cycloaddition reaction of indoles with tosyl azide, subsequent dehydroaromatization and ring-opening cascade: a computational study. Theor Chem Acc 2020;139. [DOI: 10.1007/s00214-020-02653-5] [Cited by in Crossref: 8] [Cited by in F6Publishing: 7] [Article Influence: 2.7] [Reference Citation Analysis]
|
| 10 |
Dmitriev V, Vedekhina T, Sapegin A, Krasavin M. Convenient Assembly of Privileged (Hetero)Arene‐Fused Benzo[1.4]oxazepines via Two Tandem S N Ar Events. Part 3 – (Hetero)arene‐Fused benzo[ f ]imidazo[1,2‐ d ][1,4]oxazepines. ChemistrySelect 2020;5:7873-7879. [DOI: 10.1002/slct.202002033] [Cited by in Crossref: 2] [Cited by in F6Publishing: 2] [Article Influence: 0.7] [Reference Citation Analysis]
|
| 11 |
Suryapeta S, Papigani N, Banothu V, Dubey PK, Mukkanti K, Pal S. Synthesis, biological evaluation, and docking study of a series of 1,4‐disubstituted 1,2,3‐triazole derivatives with an indole‐triazole‐peptide conjugate. J Heterocyclic Chem 2020;57:3126-41. [DOI: 10.1002/jhet.4020] [Cited by in Crossref: 11] [Cited by in F6Publishing: 13] [Article Influence: 3.7] [Reference Citation Analysis]
|
| 12 |
Bakholdina A, Lukin A, Bakulina O, Guranova N, Krasavin M. Dual use of propargylamine building blocks in the construction of polyheterocyclic scaffolds. Tetrahedron Letters 2020;61:151970. [DOI: 10.1016/j.tetlet.2020.151970] [Cited by in Crossref: 1] [Article Influence: 0.3] [Reference Citation Analysis]
|
| 13 |
Arjunan V, Durgadevi G, Mohan S. An experimental and theoretical investigation on the structure, vibrations and reactivity properties of pharmacologically active compounds 3–acetylindole and indole–3–acetamide. Journal of Molecular Structure 2020;1210:128012. [DOI: 10.1016/j.molstruc.2020.128012] [Cited by in Crossref: 5] [Article Influence: 1.7] [Reference Citation Analysis]
|
| 14 |
Zhou D. DFT investigation on the mechanism of catalytic reaction between 3-diazoindolin-2-imines and N-ethylaniline catalyzed by Rh2(Oct)4. Chemical Physics 2020;531:110661. [DOI: 10.1016/j.chemphys.2019.110661] [Cited by in Crossref: 10] [Cited by in F6Publishing: 10] [Article Influence: 3.3] [Reference Citation Analysis]
|
| 15 |
Vedekhina T, Lukin A, Krasavin M. Unexpected outcome of the Zn(OTf)2-catalyzed arylhydrazination of alkanoyl propargylamines: Rapid entry into 1-(arylamino)imidazoles. Tetrahedron Letters 2020;61:151365. [DOI: 10.1016/j.tetlet.2019.151365] [Cited by in Crossref: 1] [Cited by in F6Publishing: 1] [Article Influence: 0.3] [Reference Citation Analysis]
|
| 16 |
Vedekhina T, Lukin A, Rogacheva E, Kraeva L, Krasavin M. Zn(OTf)2-catalyzed arenehydrazination of protected propargylamines leading to 3-amidoindoles. Tetrahedron Letters 2020;61:151430. [DOI: 10.1016/j.tetlet.2019.151430] [Cited by in Crossref: 2] [Cited by in F6Publishing: 2] [Article Influence: 0.7] [Reference Citation Analysis]
|
| 17 |
Zhang G, Lin L, Yang K, Wang S, Feng Q, Zhu J, Song Q. 3‐Aminoindole Synthesis from 2‐Nitrochalcones and Ammonia or Primary Amines. Adv Synth Catal 2019;361:3718-22. [DOI: 10.1002/adsc.201900551] [Cited by in Crossref: 9] [Cited by in F6Publishing: 9] [Article Influence: 2.3] [Reference Citation Analysis]
|
| 18 |
Diao P, Hu M, Yang H, You W, Zhao P. Facile one-pot synthesis, antiproliferative evaluation and structure-activity relationships of 3-amino-1H-indoles and 3-amino-1H-7-azaindoles. Bioorganic Chemistry 2019;88:102914. [DOI: 10.1016/j.bioorg.2019.04.008] [Cited by in Crossref: 6] [Cited by in F6Publishing: 6] [Article Influence: 1.5] [Reference Citation Analysis]
|
| 19 |
Lukin A, Bakholdina A, Kryukova A, Sapegin A, Krasavin M. A three-component, Zn(OTf)2-mediated entry into trisubstituted 2-aminoimidazoles. Beilstein J Org Chem 2019;15:1061-4. [PMID: 31164943 DOI: 10.3762/bjoc.15.103] [Cited by in Crossref: 4] [Cited by in F6Publishing: 4] [Article Influence: 1.0] [Reference Citation Analysis]
|
| 20 |
Watanabe K, Moriyama K. Cu-Catalyzed Oxidative 3-Amination of Indoles via Formation of Indolyl(aryl)iodonium Imides Using o-Substituted (Diacetoxyiodo)arene as a High-Performance Hypervalent Iodine Compound. Molecules 2019;24:E1147. [PMID: 30909483 DOI: 10.3390/molecules24061147] [Cited by in Crossref: 2] [Cited by in F6Publishing: 3] [Article Influence: 0.5] [Reference Citation Analysis]
|
| 21 |
Safrygin A, Dar'in D, Lukin A, Bakholdina A, Sapegin A, Krasavin M. Zn(OTf)2-catalyzed, microwave-promoted synthesis of 2-substituted 5-methyloxazoles from propargylic amides. Tetrahedron Letters 2019;60:777-9. [DOI: 10.1016/j.tetlet.2019.02.011] [Cited by in Crossref: 9] [Cited by in F6Publishing: 9] [Article Influence: 2.3] [Reference Citation Analysis]
|
| 22 |
Leijendekker LH, Weweler J, Leuther TM, Kratzert D, Streuff J. Development, Scope, and Applications of Titanium(III)-Catalyzed Cyclizations to Aminated N-Heterocycles. Chem Eur J 2019;25:3382-90. [DOI: 10.1002/chem.201805909] [Cited by in Crossref: 17] [Cited by in F6Publishing: 17] [Article Influence: 4.3] [Reference Citation Analysis]
|
| 23 |
Watanabe K, Moriyama K. Copper-Catalyzed Indole-Selective C-N Coupling Reaction of Indolyl(2-alkoxy-phenyl)iodonium Imides: Effect of Substituent on Iodoarene as Dummy Ligand. J Org Chem 2018;83:14827-33. [PMID: 30371085 DOI: 10.1021/acs.joc.8b02676] [Cited by in Crossref: 7] [Cited by in F6Publishing: 7] [Article Influence: 1.4] [Reference Citation Analysis]
|
| 24 |
Lauder K, Toscani A, Scalacci N, Castagnolo D. Synthesis and Reactivity of Propargylamines in Organic Chemistry. Chem Rev 2017;117:14091-200. [PMID: 29166000 DOI: 10.1021/acs.chemrev.7b00343] [Cited by in Crossref: 246] [Cited by in F6Publishing: 259] [Article Influence: 41.0] [Reference Citation Analysis]
|
| 25 |
Ortiz GX Jr, Hemric BN, Wang Q. Direct and Selective 3-Amidation of Indoles Using Electrophilic N-[(Benzenesulfonyl)oxy]amides. Org Lett 2017;19:1314-7. [PMID: 28281340 DOI: 10.1021/acs.orglett.7b00358] [Cited by in Crossref: 23] [Cited by in F6Publishing: 24] [Article Influence: 3.8] [Reference Citation Analysis]
|
| 26 |
Fischer Indole Synthesis. Indole Ring Synthesis 2016. [DOI: 10.1002/9781118695692.ch2] [Cited by in F6Publishing: 1] [Reference Citation Analysis]
|
| 27 |
Zhou D, Zhou P, Jing H. Mechanisms of cascade reactions between N-methylindole and sulfonylazides via Huisgen cycloaddition: A theoretical investigation. Journal of Molecular Catalysis A: Chemical 2016;417:19-27. [DOI: 10.1016/j.molcata.2016.03.010] [Cited by in Crossref: 5] [Cited by in F6Publishing: 5] [Article Influence: 0.7] [Reference Citation Analysis]
|
| 28 |
Hu Z, Tong X, Liu G. Rhodium(III)-Catalyzed Cascade Cyclization/Electrophilic Amidation for the Synthesis of 3-Amidoindoles and 3-Amidofurans. Org Lett 2016;18:2058-61. [DOI: 10.1021/acs.orglett.6b00689] [Cited by in Crossref: 39] [Cited by in F6Publishing: 42] [Article Influence: 5.6] [Reference Citation Analysis]
|
| 29 |
Lukin A, Vedekhina T, Tovpeko D, Zhurilo N, Krasavin M. Zn-catalyzed hydrohydrazination of propargylamides with BocNHNH 2 : a novel entry into the 1,2,4-triazine core. RSC Adv 2016;6:57956-9. [DOI: 10.1039/c6ra12664b] [Cited by in Crossref: 15] [Cited by in F6Publishing: 15] [Article Influence: 2.1] [Reference Citation Analysis]
|
| 30 |
Sheng G, Huang K, Chi Z, Ding H, Xing Y, Lu P, Wang Y. Preparation of 3-Diazoindolin-2-imines via Cascade Reaction between Indoles and Sulfonylazides and Their Extensions to 2,3-Diaminoindoles and Imidazo[4,5- b ]indoles. Org Lett 2014;16:5096-9. [DOI: 10.1021/ol502423k] [Cited by in Crossref: 77] [Cited by in F6Publishing: 77] [Article Influence: 8.6] [Reference Citation Analysis]
|
| 31 |
Sharif M, Pews-davtyan A, Lukas J, Pohlers S, Rolfs A, Langer P, Beller M. Palladium-catalysed Suzuki–Miyaura coupling reactions of Bromhexine and Ambroxol. Tetrahedron 2014;70:5128-35. [DOI: 10.1016/j.tet.2014.05.116] [Cited by in Crossref: 9] [Cited by in F6Publishing: 9] [Article Influence: 1.0] [Reference Citation Analysis]
|
| 32 |
Miyata O, Ueda M, Ito Y, Matsuda N, Nishida Y. Sequential Radical Addition and Fischer-Type Indolization Reactions of Conjugated Hydrazones for the Preparation of α-Alkylindole-3-acetic Acids. HETEROCYCLES 2014;89:963. [DOI: 10.3987/com-14-12957] [Cited by in Crossref: 3] [Cited by in F6Publishing: 3] [Article Influence: 0.3] [Reference Citation Analysis]
|
| 33 |
Saito T, Sonoki Y, Otani T, Kutsumura N. Triflic acid-promoted cycloisomerization of 2-alkynylphenyl isothiocyanates and isocyanates: a novel synthetic method for a variety of indole derivatives. Org Biomol Chem 2014;12:8398-407. [DOI: 10.1039/c4ob00825a] [Cited by in Crossref: 21] [Cited by in F6Publishing: 20] [Article Influence: 2.3] [Reference Citation Analysis]
|
| 34 |
Sharif M, Pews-davtyan A, Lukas J, Schranck J, Langer P, Rolfs A, Beller M. Palladium-Catalyzed Carbonylative Transformations of Bromhexine into Bioactive Compounds as Glucocerebrosidase Inhibitors: Palladium-Catalyzed Carbonylative Transformations of Bromhexine. Eur J Org Chem 2014;2014:222-30. [DOI: 10.1002/ejoc.201301180] [Cited by in Crossref: 11] [Cited by in F6Publishing: 11] [Article Influence: 1.1] [Reference Citation Analysis]
|
| 35 |
Fukumoto Y, Ohmae A, Hirano M, Chatani N. Rhodium-Catalyzed Anti-Markovnikov Hydrohydrazination of Terminal Alkynes with N -Alkyl- and N , N -Dialkylhydrazines. Asian Journal of Organic Chemistry 2013;2:1036-9. [DOI: 10.1002/ajoc.201300188] [Cited by in Crossref: 9] [Cited by in F6Publishing: 10] [Article Influence: 0.9] [Reference Citation Analysis]
|
| 36 |
Xu M, Xu K, Wang S, Yao Z. Assembly of indolo[1,2-c]quinazolines using ZnBr2-promoted domino hydroamination–cyclization. Tetrahedron Letters 2013;54:4675-8. [DOI: 10.1016/j.tetlet.2013.06.079] [Cited by in Crossref: 24] [Cited by in F6Publishing: 24] [Article Influence: 2.4] [Reference Citation Analysis]
|
| 37 |
Bandini M. Electrophilicity: the “dark-side” of indole chemistry. Org Biomol Chem 2013;11:5206. [DOI: 10.1039/c3ob40735g] [Cited by in Crossref: 109] [Cited by in F6Publishing: 109] [Article Influence: 10.9] [Reference Citation Analysis]
|
| 38 |
Eisenlöffel C, Schmöle AC, Pews-Davtyan A, Brennführer A, Kuznetsov SA, Hübner R, Frech S, Schult C, Junghanss C, Beller M, Rolfs A, Frech MJ. Interference of a novel indolylmaleimide with microtubules induces mitotic arrest and apoptosis in human progenitor and cancer cells. Biochem Pharmacol 2013;85:763-71. [PMID: 23274302 DOI: 10.1016/j.bcp.2012.12.013] [Cited by in Crossref: 10] [Cited by in F6Publishing: 11] [Article Influence: 0.9] [Reference Citation Analysis]
|
| 39 |
Yao B, Wang Q, Zhu J. Palladium(II)-Catalyzed Intramolecular Diamination of Alkynes under Aerobic Oxidative Conditions: Catalytic Turnover of an Iodide Ion. Angew Chem Int Ed 2012;51:5170-4. [DOI: 10.1002/anie.201201640] [Cited by in Crossref: 137] [Cited by in F6Publishing: 137] [Article Influence: 12.5] [Reference Citation Analysis]
|
| 40 |
Yao B, Wang Q, Zhu J. Palladium(II)-Catalyzed Intramolecular Diamination of Alkynes under Aerobic Oxidative Conditions: Catalytic Turnover of an Iodide Ion. Angew Chem 2012;124:5260-4. [DOI: 10.1002/ange.201201640] [Cited by in Crossref: 46] [Cited by in F6Publishing: 46] [Article Influence: 4.2] [Reference Citation Analysis]
|
| 41 |
Neue B, Reiermann R, Gerdes K, Fröhlich R, Wibbeling B, Würthwein EU. Ring closure reactions of 2,6-diazaheptatrienyl metal compounds: synthesis of 3-aminoindole derivatives and 14-membered macrocyclic dimers. J Org Chem 2011;76:8794-806. [PMID: 21988327 DOI: 10.1021/jo201521v] [Cited by in Crossref: 8] [Cited by in F6Publishing: 8] [Article Influence: 0.7] [Reference Citation Analysis]
|
| 42 |
Çelebi-Ölçüm N, Boal BW, Huters AD, Garg NK, Houk KN. Why do some Fischer indolizations fail? J Am Chem Soc 2011;133:5752-5. [PMID: 21443189 DOI: 10.1021/ja201035b] [Cited by in Crossref: 49] [Cited by in F6Publishing: 50] [Article Influence: 4.1] [Reference Citation Analysis]
|
| 43 |
Benkovics T, Guzei IA, Yoon TP. Oxaziridine-mediated oxyamination of indoles: an approach to 3-aminoindoles and enantiomerically enriched 3-aminopyrroloindolines. Angew Chem Int Ed Engl 2010;49:9153-7. [PMID: 20967810 DOI: 10.1002/anie.201004635] [Cited by in Crossref: 106] [Cited by in F6Publishing: 107] [Article Influence: 8.8] [Reference Citation Analysis]
|
| 44 |
Pews-davtyan A, Beller M. Efficient and simple zinc-mediated synthesis of 3-amidoindoles. Org Biomol Chem 2011;9:6331. [DOI: 10.1039/c1ob05576c] [Cited by in Crossref: 29] [Cited by in F6Publishing: 29] [Article Influence: 2.4] [Reference Citation Analysis]
|
| 45 |
Patil NT, Singh V. Alkyne hydroamination triggered cyclizations: A powerful tool for the construction of biologically important structural motifs. Journal of Organometallic Chemistry 2011;696:419-32. [DOI: 10.1016/j.jorganchem.2010.10.027] [Cited by in Crossref: 76] [Cited by in F6Publishing: 74] [Article Influence: 6.3] [Reference Citation Analysis]
|
| 46 |
Gruit M, Pews-davtyan A, Beller M. Platinum-catalyzed cyclization reaction of alkynes: synthesis of azepino[3,4-b]indol-1-ones. Org Biomol Chem 2011;9:1148-59. [DOI: 10.1039/c0ob00728e] [Cited by in Crossref: 39] [Cited by in F6Publishing: 39] [Article Influence: 3.3] [Reference Citation Analysis]
|
| 47 |
Russel JS, Pelkey ET, Greger JG. Five-Membered Ring Systems. Elsevier; 2011. pp. 155-94. [DOI: 10.1016/b978-0-08-096805-6.00006-1] [Cited by in Crossref: 8] [Article Influence: 0.7] [Reference Citation Analysis]
|
| 48 |
Pews-davtyan A, Beller M. A novel Zn-catalyzed hydroamination of propargylamides: a general synthesis of di- and tri-substituted imidazoles. Chem Commun 2011;47:2152. [DOI: 10.1039/c0cc04625f] [Cited by in Crossref: 37] [Cited by in F6Publishing: 37] [Article Influence: 3.1] [Reference Citation Analysis]
|
| 49 |
Ortinau S, Schmich J, Block S, Liedmann A, Jonas L, Weiss DG, Helm CA, Rolfs A, Frech MJ. Effect of 3D-scaffold formation on differentiation and survival in human neural progenitor cells. Biomed Eng Online 2010;9:70. [PMID: 21070668 DOI: 10.1186/1475-925X-9-70] [Cited by in Crossref: 58] [Cited by in F6Publishing: 61] [Article Influence: 4.5] [Reference Citation Analysis]
|
| 50 |
Patil NT, Konala A. Mechanistic Dichotomy with Alkynes in the Formal Hydrohydrazination/Fischer Indolization Tandem Reaction Catalyzed by a Ph3PAuNTf2/pTSA Binary System. Eur J Org Chem 2010;2010:6831-9. [DOI: 10.1002/ejoc.201001114] [Cited by in Crossref: 40] [Cited by in F6Publishing: 40] [Article Influence: 3.1] [Reference Citation Analysis]
|
| 51 |
Benkovics T, Guzei IA, Yoon TP. Oxaziridine-Mediated Oxyamination of Indoles: An Approach to 3-Aminoindoles and Enantiomerically Enriched 3-Aminopyrroloindolines. Angewandte Chemie 2010;122:9339-43. [DOI: 10.1002/ange.201004635] [Cited by in Crossref: 27] [Cited by in F6Publishing: 27] [Article Influence: 2.1] [Reference Citation Analysis]
|
| 52 |
Pews-davtyan A, Tillack A, Schmoele A, Ortinau S, Frech MJ, Rolfs A, Beller M. ChemInform Abstract: A New Facile Synthesis of 3-Amidoindole Derivatives and Their Evaluation as Potential GSK-3β Inhibitors. ChemInform 2010;41:no-no. [DOI: 10.1002/chin.201027106] [Reference Citation Analysis]
|
