BPG is committed to discovery and dissemination of knowledge
Cited by in F6Publishing
For: Ghosh AK, Brindisi M. Urea Derivatives in Modern Drug Discovery and Medicinal Chemistry. J Med Chem 2020;63:2751-88. [PMID: 31789518 DOI: 10.1021/acs.jmedchem.9b01541] [Cited by in Crossref: 41] [Cited by in F6Publishing: 23] [Article Influence: 13.7] [Reference Citation Analysis]
Number Citing Articles
1 Efeoglu C, Yetkin D, Nural Y, Ece A, Seferoğlu Z, Ayaz F. Novel urea-thiourea hybrids bearing 1,4-naphthoquinone moiety: Anti-inflammatory activity on mammalian macrophages by regulating intracellular PI3K pathway, and molecular docking study. Journal of Molecular Structure 2022;1264:133284. [DOI: 10.1016/j.molstruc.2022.133284] [Reference Citation Analysis]
2 Greco F, Falanga AP, Terracciano M, D’ambrosio C, Piccialli G, Oliviero G, Roviello GN, Borbone N. CD, UV, and In Silico Insights on the Effect of 1,3-Bis(1′-uracilyl)-2-propanone on Serum Albumin Structure. Biomolecules 2022;12:1071. [DOI: 10.3390/biom12081071] [Reference Citation Analysis]
3 Keleş Atıcı R, Doğan ŞD, Gündüz MG, Krishna VS, Chebaiki M, Homberset H, Lherbet C, Mourey L, Tønjum T. Urea derivatives carrying a thiophenylthiazole moiety: Design, synthesis, and evaluation of antitubercular and InhA inhibitory activities. Drug Dev Res 2022. [PMID: 35769019 DOI: 10.1002/ddr.21958] [Reference Citation Analysis]
4 Xie W, Wang M, Yang S, Chen Y, Feng J, Huang Y. C-H chlorination of (hetero)anilines via photo/organo co-catalysis. Org Biomol Chem 2022. [PMID: 35730736 DOI: 10.1039/d2ob00834c] [Reference Citation Analysis]
5 Motahari R, Boshagh MA, Moghimi S, Peytam F, Hasanvand Z, Oghabi Bakhshaiesh T, Foroumadi R, Bijanzadeh H, Firoozpour L, Khalaj A, Esmaeili R, Foroumadi A. Design, synthesis and evaluation of novel tetrahydropyridothienopyrimidin-ureas as cytotoxic and anti-angiogenic agents. Sci Rep 2022;12:9683. [PMID: 35690595 DOI: 10.1038/s41598-022-13515-4] [Reference Citation Analysis]
6 Babin V, Sallustrau A, Molins M, Labiche A, Goudet A, Taran F, Audisio D. Parallel Screening with 14 C‐Labeled Carbon Dioxide: De‐risking the Staudinger‐Aza‐Wittig Reaction**. European J Organic Chem. [DOI: 10.1002/ejoc.202200133] [Reference Citation Analysis]
7 Babin V, Taran F, Audisio D. Late-Stage Carbon-14 Labeling and Isotope Exchange: Emerging Opportunities and Future Challenges. JACS Au. [DOI: 10.1021/jacsau.2c00030] [Reference Citation Analysis]
8 Pushpakumar K, Varalakshmi M, Sankar AUR, Naidu RM, Umamahesh K, Reddy DV, Raju CN. Synthesis, Spectral Characterization, and Antimicrobial Evaluation of N,N′-(1,4-Phenylene)diurea Derivatives. Russ J Org Chem 2022;58:612-8. [DOI: 10.1134/s1070428022040212] [Reference Citation Analysis]
9 Satheeshkumar R, Prabha K, Vennila KN, Sayin K, Güney E, Kaminsky W, Acevedo R. Spectroscopic (FT-IR, NMR, single crystal XRD) and DFT studies including FMO, Mulliken charges, and Hirshfeld surface analysis, molecular docking and ADME analyses of 2-amino-4′-fluorobenzophenone (FAB). Journal of Molecular Structure 2022. [DOI: 10.1016/j.molstruc.2022.133552] [Reference Citation Analysis]
10 Owen AE, Preiss A, Mcluskie A, Gao C, Peters G, Bühl M, Kumar A. Manganese-Catalyzed Dehydrogenative Synthesis of Urea Derivatives and Polyureas. ACS Catal . [DOI: 10.1021/acscatal.2c00850] [Reference Citation Analysis]
11 Njikan S, Ahmed S, Manning A, Awasthi D, Ovechkina Y, Chowdhury S, Butts A, Parish T. Chemical Exploration of a Highly Selective Scaffold with Activity against Intracellular Mycobacterium tuberculosis. Microbiol Spectr 2022;:e0116122. [PMID: 35612308 DOI: 10.1128/spectrum.01161-22] [Reference Citation Analysis]
12 Qaroush AK, Alsayyed AW, Eftaiha AF, Al‐qaisi FM, Salameh BA. Green Microwave‐Assisted Synthesis of Cyclic/Acyclic Ureas from Propylene Carbonate. ChemistrySelect 2022;7. [DOI: 10.1002/slct.202200478] [Cited by in Crossref: 1] [Cited by in F6Publishing: 1] [Article Influence: 1.0] [Reference Citation Analysis]
13 Bhosle SD, Itage SV, Jadhav KA, Eppa G, Bhosale RS, Yadav JS. Zn Mediated Urea Bond Formation: A Novel and Convenient Method. ChemistrySelect 2022;7. [DOI: 10.1002/slct.202201004] [Reference Citation Analysis]
14 Ahmad S, Ahmad HW, Bhatt P. Microbial adaptation and impact into the pesticide's degradation. Arch Microbiol 2022;204:288. [PMID: 35482163 DOI: 10.1007/s00203-022-02899-6] [Reference Citation Analysis]
15 Chakrabortty P, Biswas S, Das A, Dolai M, Islam SM. Diformylphloroglucinol derived imine based covalent organic frameworks (PHTA) as efficient organocatalyst for conversion of isocyanates to urea derivatives. Molecular Catalysis 2022;522:112213. [DOI: 10.1016/j.mcat.2022.112213] [Reference Citation Analysis]
16 Feng Y, Zhang B, Lv J, Zhang P, Mao Q, Lin F, Zhao J, Fu X, Yang Y, Li Z, Zhang L, Mou Y, Wang S. Scaffold hopping of celastrol provides derivatives containing pepper ring, pyrazine and oxazole substructures as potent autophagy inducers against breast cancer cell line MCF-7. European Journal of Medicinal Chemistry 2022;234:114254. [DOI: 10.1016/j.ejmech.2022.114254] [Reference Citation Analysis]
17 Sochacka-Ćwikła A, Mączyński M, Regiec A. FDA-Approved Small Molecule Compounds as Drugs for Solid Cancers from Early 2011 to the End of 2021. Molecules 2022;27:2259. [PMID: 35408658 DOI: 10.3390/molecules27072259] [Reference Citation Analysis]
18 Bouayad-Gervais S, Nielsen CD, Turksoy A, Sperger T, Deckers K, Schoenebeck F. Access to Cyclic N-Trifluoromethyl Ureas through Photocatalytic Activation of Carbamoyl Azides. J Am Chem Soc 2022. [PMID: 35333063 DOI: 10.1021/jacs.2c02004] [Reference Citation Analysis]
19 Kasatkina SO, Geyl KK, Baykov SV, Novikov MS, Boyarskiy VP. “Urea to Urea” Approach: Access to Unsymmetrical Ureas Bearing Pyridyl Substituents. Adv Synth Catal 2022;364:1295-304. [DOI: 10.1002/adsc.202101490] [Reference Citation Analysis]
20 Wu J, Zhu RD, Cao GM, Du JC, Liu X, Diao LZ, Zhang ZY, Hu YS, Liu XH, Shi JB. Discovery of novel paeonol-based derivatives against skin inflammation in vitro and in vivo. Journal of Enzyme Inhibition and Medicinal Chemistry 2022;37:817-31. [DOI: 10.1080/14756366.2022.2043852] [Reference Citation Analysis]
21 Firooz SK, Putman J, Fulton B, Lovely CJ, Berthod A, Armstrong DW. Liquid chromatography enantiomeric separation of chiral ethanolamine substituted compounds. Chirality. [DOI: 10.1002/chir.23419] [Reference Citation Analysis]
22 Law CSW, Yeong KY. Current trends of benzothiazoles in drug discovery: a patent review (2015–2020). Expert Opinion on Therapeutic Patents. [DOI: 10.1080/13543776.2022.2026327] [Reference Citation Analysis]
23 Baeva LA, Biktasheva LF, Nugumanov TR, Fatykhov AA. Multicomponent Synthesis of 1,3-Bis[(alkylsulfanyl)methyl]-1,3,5-triazinan-2-ones. Russ J Org Chem 2021;57:1948-54. [DOI: 10.1134/s1070428021120071] [Reference Citation Analysis]
24 D'agostino I, Ardino C, Poli G, Sannio F, Lucidi M, Poggialini F, Visaggio D, Rango E, Filippi S, Petricci E, Visca P, Botta L, Docquier J, Dreassi E. Antibacterial alkylguanidino ureas: Molecular simplification approach, searching for membrane-based MoA. European Journal of Medicinal Chemistry 2022. [DOI: 10.1016/j.ejmech.2022.114158] [Cited by in Crossref: 1] [Article Influence: 1.0] [Reference Citation Analysis]
25 Yang Z, Zhou Z, Luo X, Luo X, Luo H, Luo L, Yang W. Design and Synthesis of Novel Podophyllotoxins Hybrids and the Effects of Different Functional Groups on Cytotoxicity. Molecules 2021;27:220. [PMID: 35011453 DOI: 10.3390/molecules27010220] [Reference Citation Analysis]
26 Vannozzi G, Vullo D, Angeli A, Ferraroni M, Combs J, Lomelino C, Andring J, Mckenna R, Bartolucci G, Pallecchi M, Lucarini L, Sgambellone S, Masini E, Carta F, Supuran CT. One-Pot Procedure for the Synthesis of Asymmetric Substituted Ureido Benzene Sulfonamides as Effective Inhibitors of Carbonic Anhydrase Enzymes. J Med Chem 2021. [PMID: 34958217 DOI: 10.1021/acs.jmedchem.1c01906] [Reference Citation Analysis]
27 Salam R, Chowdhury SM, Marshall SR, Gneid H, Busschaert N. Increasing membrane permeability of carboxylic acid-containing drugs using synthetic transmembrane anion transporters. Chem Commun (Camb) 2021;57:13122-5. [PMID: 34783329 DOI: 10.1039/d1cc02327f] [Reference Citation Analysis]
28 Dombrowski AW, Aguirre AL, Shrestha A, Sarris KA, Wang Y. The Chosen Few: Parallel Library Reaction Methodologies for Drug Discovery. J Org Chem 2021. [PMID: 34780177 DOI: 10.1021/acs.joc.1c01427] [Cited by in Crossref: 1] [Cited by in F6Publishing: 1] [Article Influence: 1.0] [Reference Citation Analysis]
29 Song X, Liu X, Yu W, Jin Y. Amide-Assisted Rearrangement of Hydroxyarylformimidoyl Chloride to Diarylurea. Molecules 2021;26:6437. [PMID: 34770846 DOI: 10.3390/molecules26216437] [Reference Citation Analysis]
30 Poonia N, Lal K, Kumar A, Kumar A, Sahu S, Baidya ATK, Kumar R. Urea-thiazole/benzothiazole hybrids with a triazole linker: synthesis, antimicrobial potential, pharmacokinetic profile and in silico mechanistic studies. Mol Divers 2021. [PMID: 34671895 DOI: 10.1007/s11030-021-10336-x] [Reference Citation Analysis]
31 Lan CB, Auclair K. Ammonium Chloride‐Promoted Rapid Synthesis of Monosubstituted Ureas under Microwave Irradiation. Eur J Org Chem 2021;2021:5135-46. [DOI: 10.1002/ejoc.202101059] [Cited by in Crossref: 1] [Cited by in F6Publishing: 1] [Article Influence: 1.0] [Reference Citation Analysis]
32 Shafiei M, Toreyhi H, Firoozpour L, Akbarzadeh T, Amini M, Hosseinzadeh E, Hashemzadeh M, Peyton L, Lotfali E, Foroumadi A. Design, Synthesis, and In Vitro and In Vivo Evaluation of Novel Fluconazole-Based Compounds with Promising Antifungal Activities. ACS Omega 2021;6:24981-5001. [PMID: 34604679 DOI: 10.1021/acsomega.1c04016] [Cited by in Crossref: 1] [Cited by in F6Publishing: 1] [Article Influence: 1.0] [Reference Citation Analysis]
33 Yu M, Li C, He M, Zhu Y, Yang R, Deng S, Meng X, Yao R. Structure–activity relationship studies on Pd176252 derivatives leading to discovery of novel GRP receptor antagonist with potent anticancer activity. Med Chem Res. [DOI: 10.1007/s00044-021-02793-8] [Reference Citation Analysis]
34 Singh DK, Chauthe SK, Anjanappa P, Kumar S, Arulraj RA, Gajjela R, Mohammed N, Kanthappa VT, Karmakar A, Gupta AK, Bajpai L, Bagadi M, Mathur A. Synthesis and characterization of a series of N,N'-substituted urea derivatives by using electrospray ionization tandem mass spectrometry: Differentiation of positional isomers. Rapid Commun Mass Spectrom 2021;35:e9161. [PMID: 34240514 DOI: 10.1002/rcm.9161] [Reference Citation Analysis]
35 Babin V, Sallustrau A, Loreau O, Caillé F, Goudet A, Cahuzac H, Del Vecchio A, Taran F, Audisio D. A general procedure for carbon isotope labeling of linear urea derivatives with carbon dioxide. Chem Commun (Camb) 2021;57:6680-3. [PMID: 34132265 DOI: 10.1039/d1cc02665h] [Reference Citation Analysis]
36 Jakobsson JE, Telu S, Lu S, Jana S, Pike VW. Broad Scope and High-Yield Access to Unsymmetrical Acyclic [11 C]Ureas for Biomedical Imaging from [11 C]Carbonyl Difluoride. Chemistry 2021;27:10369-76. [PMID: 33890705 DOI: 10.1002/chem.202100690] [Cited by in Crossref: 1] [Cited by in F6Publishing: 1] [Article Influence: 1.0] [Reference Citation Analysis]
37 Kuznetsov YP, Degtyarenko EK, Burmistrov VV, Saeef MHA, Pitushkin DA, Vernigora AA, Butov GM. Synthesis and Properties of N,N′-Disubstituted Ureas and Their Isosteric Analogs Containing Polycyclic Fragments: IX. N-(1,7,7-Trimethylbicyclo[2.2.1]heptan-2-yl) Ureas and Thioureas. Russ J Org Chem 2021;57:515-23. [DOI: 10.1134/s1070428021040035] [Cited by in Crossref: 2] [Cited by in F6Publishing: 1] [Article Influence: 2.0] [Reference Citation Analysis]
38 Petti A, Fagnan C, van Melis CGW, Tanbouza N, Garcia AD, Mastrodonato A, Leech MC, Goodall ICA, Dobbs AP, Ollevier T, Lam K. Supporting-Electrolyte-Free Anodic Oxidation of Oxamic Acids into Isocyanates: An Expedient Way to Access Ureas, Carbamates, and Thiocarbamates. Org Process Res Dev 2021;25:2614-21. [DOI: 10.1021/acs.oprd.1c00112] [Cited by in Crossref: 2] [Cited by in F6Publishing: 1] [Article Influence: 2.0] [Reference Citation Analysis]
39 Ronchetti R, Moroni G, Carotti A, Gioiello A, Camaioni E. Recent advances in urea- and thiourea-containing compounds: focus on innovative approaches in medicinal chemistry and organic synthesis. RSC Med Chem 2021;12:1046-64. [PMID: 34355177 DOI: 10.1039/d1md00058f] [Reference Citation Analysis]
40 Watson RB, Butler TW, Deforest JC. Preparation of Carbamates, Esters, Amides, and Unsymmetrical Ureas via Brønsted Acid-Activated N -Acyl Imidazoliums. Org Process Res Dev 2021;25:500-6. [DOI: 10.1021/acs.oprd.0c00445] [Cited by in Crossref: 1] [Cited by in F6Publishing: 1] [Article Influence: 1.0] [Reference Citation Analysis]
41 Mandal S, Pramanik A. Three-Component Synthesis of Pyrrolo/indolo[1,2- a ]quinoxalines Substituted with o -Biphenylester/ N -arylcarbamate/ N -arylurea: A Domino Approach Involving Spirocyclic Ring Opening. J Org Chem 2021;86:5047-64. [DOI: 10.1021/acs.joc.0c02973] [Cited by in Crossref: 2] [Cited by in F6Publishing: 2] [Article Influence: 2.0] [Reference Citation Analysis]
42 Li C, Zhong J, Liu B, Yang T, Lv B, Luo Y. Study on Typical Diarylurea Drugs or Derivatives in Cocrystallizing with Strong H-Bond Acceptor DMSO. ACS Omega 2021;6:5532-47. [PMID: 33681594 DOI: 10.1021/acsomega.0c05908] [Reference Citation Analysis]
43 Pitushkin DA, Burmistrov VV, Kuznetsov YP, Ivankina OM, Butov GM. Synthesis and Properties of N,N′-Disubstituted Ureas and Their Isosteric Analogs Containing Polycyclic Fragments: VI. N-[Fluoro(chloro)phenyl]-N′-(4,7,7-trimethyl-3-oxo-2-oxabicyclo[2.2.1]heptan-1-yl)ureas. Russ J Org Chem 2020;56:2057-66. [DOI: 10.1134/s1070428020120027] [Cited by in Crossref: 1] [Article Influence: 1.0] [Reference Citation Analysis]
44 Al-ostoot FH, Zabiulla, Salah S, Khanum SA. Recent investigations into synthesis and pharmacological activities of phenoxy acetamide and its derivatives (chalcone, indole and quinoline) as possible therapeutic candidates. J IRAN CHEM SOC 2021;18:1839-75. [DOI: 10.1007/s13738-021-02172-5] [Cited by in Crossref: 9] [Cited by in F6Publishing: 2] [Article Influence: 9.0] [Reference Citation Analysis]
45 Zhang Y, Ge X, Lu H, Li G. Catalytic Decarboxylative C-N Formation to Generate Alkyl, Alkenyl, and Aryl Amines. Angew Chem Int Ed Engl 2021;60:1845-52. [PMID: 33026167 DOI: 10.1002/anie.202010974] [Cited by in Crossref: 7] [Cited by in F6Publishing: 3] [Article Influence: 7.0] [Reference Citation Analysis]
46 Pitushkin DA, Burmistrov VV, Saeef MHA, Vernigora AA, Butov GM. Synthesis and Properties of 1,3-Disubstituted Ureas and Their Isosteric Analogs Containing Polycyclic Fragments: V. 1-(Bicyclo[2.2.1]heptan-2-yl)-3-R- and 1-(1,7,7-Tricyclo[2.2.1]heptan-2-yl)-3-R-ureas. Russ J Org Chem 2020;56:1893-904. [DOI: 10.1134/s1070428020110020] [Cited by in Crossref: 1] [Cited by in F6Publishing: 1] [Article Influence: 1.0] [Reference Citation Analysis]
47 Catalano A, Iacopetta D, Sinicropi MS, Franchini C. Diarylureas as Antitumor Agents. Applied Sciences 2021;11:374. [DOI: 10.3390/app11010374] [Cited by in Crossref: 10] [Cited by in F6Publishing: 1] [Article Influence: 10.0] [Reference Citation Analysis]
48 Matošević A, Bosak A. Carbamate group as structural motif in drugs: a review of carbamate derivatives used as therapeutic agents. Arh Hig Rada Toksikol 2020;71:285-99. [PMID: 33410773 DOI: 10.2478/aiht-2020-71-3466] [Cited by in Crossref: 1] [Cited by in F6Publishing: 2] [Article Influence: 0.5] [Reference Citation Analysis]
49 Zhang Y, Ge X, Lu H, Li G. Catalytic Decarboxylative C−N Formation to Generate Alkyl, Alkenyl, and Aryl Amines. Angew Chem 2021;133:1873-80. [DOI: 10.1002/ange.202010974] [Cited by in Crossref: 2] [Cited by in F6Publishing: 1] [Article Influence: 1.0] [Reference Citation Analysis]
50 Akgul O, Singh S, Andring JT, McKenna R, Selleri S, Carta F, Angeli A, Supuran CT. Handling drug-target selectivity: A study on ureido containing Carbonic Anhydrase inhibitors. Eur J Med Chem 2021;212:113035. [PMID: 33303238 DOI: 10.1016/j.ejmech.2020.113035] [Cited by in Crossref: 1] [Cited by in F6Publishing: 2] [Article Influence: 0.5] [Reference Citation Analysis]
51 Xu K, Zheng Y, Ye Y, Liu D, Zhang W. Desymmetrization of meso-Dicarbonatecyclohexene with β-Hydrazino Carboxylic Esters via a Pd-Catalyzed Allylic Substitution Cascade. Org Lett 2020;22:8836-41. [PMID: 33170017 DOI: 10.1021/acs.orglett.0c03211] [Reference Citation Analysis]
52 Mohammed HHH, Abbas SH, Hayallah AM, Abuo-Rahma GEA, Mostafa YA. Novel urea linked ciprofloxacin-chalcone hybrids having antiproliferative topoisomerases I/II inhibitory activities and caspases-mediated apoptosis. Bioorg Chem 2021;106:104422. [PMID: 33248713 DOI: 10.1016/j.bioorg.2020.104422] [Cited by in Crossref: 1] [Cited by in F6Publishing: 1] [Article Influence: 0.5] [Reference Citation Analysis]
53 Pattarawarapan M, Yamano D, Wiriya N, Yimklan S, Phakhodee W. Simultaneous Formation and Functionalization of Aryliminophosphoranes Using 1,3-Dihydro-1H-benzimidazol-2-ones as Precursors. J Org Chem 2020;85:13330-8. [PMID: 33006471 DOI: 10.1021/acs.joc.0c01979] [Cited by in Crossref: 1] [Article Influence: 0.5] [Reference Citation Analysis]
54 Luo G, Lin X, Li Z, Xiao M, Li X, Zhang D, Xiang H. Structure-guided modification of isoxazole-type FXR agonists: Identification of a potent and orally bioavailable FXR modulator. Eur J Med Chem 2021;209:112910. [PMID: 33049605 DOI: 10.1016/j.ejmech.2020.112910] [Cited by in Crossref: 1] [Cited by in F6Publishing: 1] [Article Influence: 0.5] [Reference Citation Analysis]
55 Farag AK, Hassan AH, Chung K, Lee J, Gil H, Lee K, Roh EJ. Diarylurea derivatives comprising 2,4-diarylpyrimidines: Discovery of novel potential anticancer agents via combined failed-ligands repurposing and molecular hybridization approaches. Bioorganic Chemistry 2020;103:104121. [DOI: 10.1016/j.bioorg.2020.104121] [Cited by in Crossref: 3] [Cited by in F6Publishing: 2] [Article Influence: 1.5] [Reference Citation Analysis]
56 Soccio M, Mazzoni R, Lucarelli C, Quattrosoldi S, Cingolani A, Fiorini M, Lotti N, Tabanelli T. Urea and Polyurea Production: An Innovative Solvent- and Catalyst-Free Approach through Catechol Carbonate. ACS Sustainable Chem Eng 2020;8:15640-50. [DOI: 10.1021/acssuschemeng.0c05177] [Cited by in Crossref: 7] [Cited by in F6Publishing: 4] [Article Influence: 3.5] [Reference Citation Analysis]
57 He Z, Wu D, Vessally E. Cross-dehydrogenative Coupling Reactions Between Formamidic C(sp2)-H and X-H (X = C, O, N) Bonds. Top Curr Chem (Cham) 2020;378:46. [PMID: 32975616 DOI: 10.1007/s41061-020-00309-3] [Cited by in Crossref: 7] [Article Influence: 3.5] [Reference Citation Analysis]
58 Ashraf-Uz-Zaman M, Shahi S, Akwii R, Sajib MS, Farshbaf MJ, Kallem RR, Putnam W, Wang W, Zhang R, Alvina K, Trippier PC, Mikelis CM, German NA. Design, synthesis and structure-activity relationship study of novel urea compounds as FGFR1 inhibitors to treat metastatic triple-negative breast cancer. Eur J Med Chem 2021;209:112866. [PMID: 33039722 DOI: 10.1016/j.ejmech.2020.112866] [Cited by in Crossref: 1] [Cited by in F6Publishing: 1] [Article Influence: 0.5] [Reference Citation Analysis]
59 Xiao J, Gao M, Sun Z, Diao Q, Wang P, Gao F. Recent advances of podophyllotoxin/epipodophyllotoxin hybrids in anticancer activity, mode of action, and structure-activity relationship: An update (2010-2020). Eur J Med Chem 2020;208:112830. [PMID: 32992133 DOI: 10.1016/j.ejmech.2020.112830] [Cited by in Crossref: 5] [Cited by in F6Publishing: 2] [Article Influence: 2.5] [Reference Citation Analysis]
60 Kumari S, Carmona AV, Tiwari AK, Trippier PC. Amide Bond Bioisosteres: Strategies, Synthesis, and Successes. J Med Chem 2020;63:12290-358. [PMID: 32686940 DOI: 10.1021/acs.jmedchem.0c00530] [Cited by in Crossref: 34] [Cited by in F6Publishing: 26] [Article Influence: 17.0] [Reference Citation Analysis]
61 Kumar R, Bidgood CL, Levrier C, Gunter JH, Nelson CC, Sadowski MC, Davis RA. Synthesis of a Unique Psammaplysin F Library and Functional Evaluation in Prostate Cancer Cells by Multiparametric Quantitative Single Cell Imaging. J Nat Prod 2020;83:2357-66. [DOI: 10.1021/acs.jnatprod.0c00121] [Cited by in Crossref: 2] [Cited by in F6Publishing: 3] [Article Influence: 1.0] [Reference Citation Analysis]
62 Wang Q, Tuinhof J, Mgimpatsang KC, Kurpiewska K, Kalinowska-Tluscik J, Dömling A. Copper-Catalyzed Modular Assembly of Polyheterocycles. J Org Chem 2020;85:9915-27. [PMID: 32615764 DOI: 10.1021/acs.joc.0c01238] [Cited by in Crossref: 2] [Cited by in F6Publishing: 1] [Article Influence: 1.0] [Reference Citation Analysis]
63 Sun N, Huang Y, Yu M, Zhao Y, Chen JA, Zhu C, Song M, Guo H, Xie Q, Wang Y. Discovery of carboxyl-containing biaryl ureas as potent RORγt inverse agonists. Eur J Med Chem 2020;202:112536. [PMID: 32698100 DOI: 10.1016/j.ejmech.2020.112536] [Cited by in Crossref: 2] [Cited by in F6Publishing: 2] [Article Influence: 1.0] [Reference Citation Analysis]
64 Terrab L, Rosenker CJ, Johnstone L, Ngo LK, Zhang L, Ware NF, Miller B, Topacio AZ, Sannino S, Brodsky JL, Wipf P. Synthesis and Selective Functionalization of Thiadiazine 1,1-Dioxides with Efficacy in a Model of Huntington's Disease. ACS Med Chem Lett 2020;11:984-90. [PMID: 32435415 DOI: 10.1021/acsmedchemlett.0c00018] [Cited by in Crossref: 2] [Cited by in F6Publishing: 2] [Article Influence: 1.0] [Reference Citation Analysis]
65 Driscoll JP, Sadlowski CM, Shah NR, Feula A. Metabolism and Bioactivation: It's Time to Expect the Unexpected. J Med Chem 2020;63:6303-14. [PMID: 32267691 DOI: 10.1021/acs.jmedchem.0c00026] [Cited by in Crossref: 6] [Cited by in F6Publishing: 6] [Article Influence: 3.0] [Reference Citation Analysis]
66 Shamanth S, Chaithra N, Gurukiran M, Mamatha M, Lokanath NK, Rangappa KS, Mantelingu K. I2-Catalyzed transformation of o-aminobenzamide to o-ureidobenzonitrile using isothiocyanates. Org Biomol Chem 2020;18:2678-84. [PMID: 32202293 DOI: 10.1039/d0ob00118j] [Cited by in Crossref: 1] [Article Influence: 0.5] [Reference Citation Analysis]